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N-[(6-chloropyridin-3-yl)methyl]-6-methyl-2-propylpyrimidin-4-amine
2-ethyl-9-[2-(1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-3-[(1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(3-methylbutyl)-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}benzene-1,3-diol
2-(dimethylamino)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(2-methylphenyl)acetamide
6-{[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-ethyl-1,2-oxazole-5-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{1-[1-(methoxymethyl)cyclobutanecarbonyl]-1,2,3,6-tetrahydropyridin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methyl-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(1H-imidazol-1-yl)butan-1-one
methyl 3-[(5-acetamidothiophen-2-yl)methyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(3-methylfuran-2-carbonyl)piperidine-3-carboxylate
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(4-methylphenyl)propanamide
4-methyl-5-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
(2S,4S)-4-amino-1-[3-(2-oxopiperidin-1-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
ethyl 1-[(3,4-dimethylphenyl)carbamoyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-amino-4-(4-hydroxy-3-methoxyphenyl)-6-(4-methylphenyl)pyridine-3-carbonitrile
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-methyl-4-(4-{[methyl(1-methylpyrrolidin-3-yl)amino]methyl}phenyl)butan-2-ol
5-{2-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-4-carboxamide
3-(hydroxymethyl)-1-(5-phenoxyfuran-2-carbonyl)piperidin-3-ol
2-ethyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]pyrimidine-5-carboxamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(2,3,4-trifluorophenyl)propanamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
1-[3-(cyclopentyloxy)phenyl]-3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methylurea
6-{[(3S,4S)-4-(dimethylamino)-3-hydroxypiperidin-1-yl]methyl}pyridine-2-carboxylic acid
2-amino-4-(5-hydroxy-2-methoxyphenyl)-6-(4-hydroxy-2-methylphenyl)pyridine-3-carbonitrile
ethyl 3-({[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]carbamoyl}amino)propanoate
N-[(3R,4S)-1-cyclobutanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-4-(trifluoromethyl)pyrimidin-2-amine
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
1,3-dimethyl-2,6-dioxo-N-(4-phenylbutan-2-yl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
N-[2-(1-methylpiperidin-3-yl)ethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
N-(3-hydroxypropyl)-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5-(4-fluorophenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
1-methyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-imidazole-2-carboxamide
3-[(3R,4S)-1-{4-[ethyl(methyl)amino]pyrimidin-2-yl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(2-chlorophenyl)methyl]-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]propanamide
methyl 4-({[(3S,5S)-5-{[2-(2H-1,3-benzodioxol-5-yl)ethyl]carbamoyl}-1-benzylpyrrolidin-3-yl]amino}methyl)benzoate
1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-benzyl-8-(2,3-dihydro-1-benzofuran-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(4aS,7aR)-1-(2-aminopyridine-4-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-4-{2-[3-(3-methylphenoxy)azetidin-1-yl]pyridine-4-carbonyl}piperazine
N-[(1-{[5-(methylcarbamoyl)furan-2-yl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]pyrrolidine-1-carboxamide