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N-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
N-[2-(diethylamino)ethyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-methyl-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-ethyl-9-(6-methylpyrimidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-(oxan-4-yl)-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazine
N-({5-[(3-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
2-cyclopropyl-9-[2-(3-hydroxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(2S,4R)-1-benzyl-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
6-(2-fluoro-5-methylphenyl)-9H-purin-2-amine
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]oxolane-3-carboxamide
N-ethyl-6-[4-(oxan-4-yl)piperazin-1-yl]pyridine-3-carboxamide
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
1-{4-[(1-methylpiperidin-3-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
3-({4-methyl-6-[4-(1,3-thiazol-2-yl)piperazin-1-yl]pyrimidin-2-yl}amino)phenol
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-[2-(1H-indol-3-yl)ethyl]piperidine-3,5-dicarboxamide
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
N-{1-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-2-(4-fluorophenyl)ethyl}-2-(dimethylamino)-N-methylacetamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(2-methoxyphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-butyl-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-(2,2-diphenylethyl)-4-(5-methylpyrazine-2-carbonyl)morpholine
4-{1-[3-(pyridin-3-yl)propyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
N-butyl-N-methyl-3-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-chloro-N-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)amino]ethyl}benzene-1-sulfonamide
2-(propan-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzoxazole-5-carboxamide
4-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}-1,4-oxazepan-6-ol
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
(3S,4S)-1-(2-ethylpyridine-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
(2S,4S,5R)-5-(3-chlorophenyl)-4-[(3-methoxypropyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
4-ethyl-N,N-dimethyl-6-{4-[(oxan-4-yl)amino]piperidin-1-yl}pyrimidin-2-amine
(1S,6R)-9-[2-(1H-indol-3-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(2-fluorophenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-[(4-fluorophenyl)methyl]-4-[5-(methoxymethyl)thiophene-2-carbonyl]morpholine
2,6-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-4-carboxamide
8-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-{5-[1-(1-methyl-1H-imidazole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-2-amine
N-methyl-N-[(6-methylquinolin-5-yl)methyl]thian-4-amine
2-(2-{[({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amino]methyl}phenoxy)ethan-1-ol
2-butyl-8-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
2-{1-[(4-ethoxyphenyl)methyl]-4-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
[(1-methyl-1H-imidazol-2-yl)methyl](prop-2-en-1-yl)(pyridin-3-ylmethyl)amine
2-methyl-5-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]phenol
N-cyclopropyl-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridin-3-ol
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
2-methyl-N-{1-[(4-methylphenyl)methyl]cyclopropyl}furan-3-carboxamide