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(1R,5R)-3-[3-(2-ethoxyethoxy)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2,4-difluorophenyl)-1-{1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl}ethyl]-N-methylpropanamide
1-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
2-methoxy-5-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)phenol
(3R,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
4-(2-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidin-2-yl}ethyl)morpholine
N-methyl-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(2-phenylethyl)piperidin-3-amine
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
2-{4-chloro-2-[1-(1H-imidazol-2-ylmethyl)-1H-1,2,3-triazol-4-yl]phenoxy}acetic acid
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(4-methyl-1,4-diazepan-1-yl)acetamide
(2E)-N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
3-[(4aR,7aS)-4-(5-methylpyrazine-2-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
5-[(dimethylamino)methyl]-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-phenylbutane-1,4-dione
4-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
1-methyl-3-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-{[4-(difluoromethoxy)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-ethyl-3-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 4-({ethyl[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]amino}methyl)-1H-pyrazole-3-carboxylate
(2,1,3-benzoxadiazol-5-ylmethyl)[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
2-(methylsulfanyl)-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
3-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyrimidin-2-amine
2-ethoxy-5-{2-[(piperidin-4-yl)amino]pyrimidin-4-yl}benzoic acid
4-chloro-5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-4-(pyridin-2-yl)piperidin-4-ol
4-(2-methoxyphenoxy)-1-(2-methylfuran-3-carbonyl)piperidine-4-carboxylic acid
1-({5-[(1-ethylpiperidin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
5-(3,6-dimethyl-1-benzofuran-2-carbonyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}phenoxy)acetic acid
benzyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(1,3-thiazol-2-ylmethyl)amine
6-[(2-hydroxyethyl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
2-[(2-methyl-1,3-oxazol-4-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[1-benzyl-5-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
(2S,4S,5R)-4-{[(4-hydroxyphenyl)methyl]carbamoyl}-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylic acid
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
N'-(3,5-dimethylphenyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]propanediamide
(2S)-N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
N-(2-methanesulfonylethyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
N,N-dimethyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-amine
N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
5-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidine-3-carboxylate
4,6-dimethyl-1-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2-dihydropyrimidin-2-one
dimethyl(2-{[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]oxy}hex-5-en-1-yl)amine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide