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7-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)thiophene-3-carboxamide
N-cyclopentyl-6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridazin-3-amine
2-(1-methylpyrrolidin-3-yl)-9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-9H-purin-2-amine
N-(carbamoylmethyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-(4-methoxybutyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-benzyl-1-(2-methoxyethyl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidine-3-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
3-[({2-[(2-chlorophenyl)methoxy]-6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)amino]-1λ6-thiolane-1,1-dione
4-methyl-2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
5-[4-(ethanesulfonyl)piperazine-1-carbonyl]-4,6-dimethyl-1,2,3,4-tetrahydropyrimidin-2-one
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-3-(3-chlorophenyl)-3-phenylpropanamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]oxane-4-carboxamide
2-(morpholin-2-yl)-1-[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
dimethyl[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(5-methylthiophen-2-yl)methyl]amino)ethyl]amine
N-({5-[(3-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
7-(cyclopropylmethyl)-2-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-6-(4-methoxyphenyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1,8-naphthyridine-3-carboxamide
methyl[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl](oxolan-3-ylmethyl)amine
(2S,4S)-4-amino-N-methyl-1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]pyrrolidine-2-carboxamide
N-ethyl-2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide
5-[3-(trifluoromethyl)phenyl]pyrimidine
4-hydroxy-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
methyl 4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
3-(furan-2-yl)-4-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-(4-fluoro-2-methoxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
N-(1-methyl-1H-1,2,3-triazol-4-yl)-4-(1H-pyrrol-1-ylmethyl)benzamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}propan-1-one
N-[1-(1H-imidazol-2-yl)ethyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
3-(2-chloropyridin-3-yl)-1-[1-(cyclohex-1-en-1-yl)ethyl]urea
2-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-(2-ethoxyphenyl)-3-oxo-3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]propanamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-[1-(3-methylbutyl)-2,4-dioxo-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
5-{1-[(2,6-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
2-(4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
1-(5-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl)pyrrolidine
8-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
2-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)quinoline-4-carboxamide
7-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 2-[2-(2-ethylpyrimidin-4-yl)-1H-imidazol-1-yl]-2-(3-methylphenyl)acetate
N-{2-[1-(cyclopentylmethyl)piperidin-3-yl]ethyl}oxane-4-carboxamide
2-chloro-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-6-methylbenzamide
1-[1-(furan-3-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
[2,2-dimethyl-3-(morpholin-4-yl)propyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine