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N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(2H-indazol-2-yl)acetamide
1-ethyl-4-(3-propoxypiperidin-1-yl)piperidine
(1R,5S,6S)-N,N-dimethyl-3-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-propyl-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,3,4-oxadiazole
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(4-hydroxyphenyl)ethan-1-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
7-cyclohexyl-2-(1,2-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(cyclohexylmethyl)-4-[2-(morpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]acetamide
({5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-{[6-({[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}amino)pyrimidin-4-yl]amino}ethan-1-ol
2-hydroxy-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-ethyl-5-(2-methanesulfonylethyl)-3-(2-methoxyethyl)-1H-1,2,4-triazole
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
N-(2-methanesulfonylethyl)-4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-amine
N-(2-fluoro-4-methylphenyl)-2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}acetamide
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)thiophene-3-carboxamide
2-(ethylamino)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-5-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-ethyl-N-propylacetamide
N-[3-(6-cyanopyridin-2-yl)phenyl]acetamide
2-{[(5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
2-(cyclopropylmethyl)-8-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-(8-methoxyquinolin-2-yl)piperazin-2-yl}ethan-1-ol
7-[(3,4-difluorophenyl)methyl]-2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
{1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
3-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)furan-2-carboxamide
2-{3,5-dimethyl-4-[(pyrrolidine-1-sulfonyl)amino]-1H-pyrazol-1-yl}acetic acid
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylacetamide
N-[(2-methoxyphenyl)methyl]-2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}acetamide
N-cyclopropyl-3-{1-[2-(thiophen-2-yl)acetyl]piperidin-3-yl}propanamide
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-5-{1-[2-(4-methoxyphenyl)ethyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
(3S,9aR)-3-benzyl-8-[(3-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-cyclopentyl-N-[2-(dimethylamino)pentyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-methyl-9-(2,3,6-trifluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-N-ethylpyridine-4-carboxamide
2-{4-[2-amino-3-cyano-6-(3-methoxyphenyl)pyridin-4-yl]phenoxy}acetamide
4-hydroxy-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-(phenoxymethyl)pyrimidine-5-carboxamide
2-{3-[4-(4-cyanophenyl)-3-oxopiperazine-1-carbonyl]phenoxy}acetamide
3-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-N-(pyridin-3-yl)benzamide
2-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-3-(thiophen-3-yl)propan-1-ol
1-(4-chlorophenyl)-N-({1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
N-[(2S)-2-aminopropyl]-2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(2-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-2-oxoethyl)piperidin-2-one
N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide