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[(3-methyl-1,2-oxazol-5-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
1-(3,4-dimethylphenyl)-N-(oxan-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[(5-methylthiophen-2-yl)methyl]-2,7-dioxo-N-(pyridin-2-ylmethyl)-1,3-diazepane-4-carboxamide
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-[4-(propan-2-yl)phenyl]-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrrolidin-2-one
N-(1H-imidazol-2-ylmethyl)-N,2-dimethyl-2-(thiophen-2-ylformamido)propanamide
[3-({[(2-ethoxypyridin-3-yl)methyl]amino}methyl)-2,4,6-trimethylphenyl]methanol
(4aR,7aS)-1-(2-methoxyethyl)-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(piperidin-1-yl)-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydropyridazin-3-one
3-({1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
N-[2-(3,5-dimethoxyphenyl)ethyl]-3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carboxamide
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-(pyridin-3-ylmethyl)piperidin-3-ol
(1S,6R)-3-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-1-(1,4-dioxan-2-ylmethyl)-1-methylurea
1-(6-methylpyridazin-3-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(hydroxymethyl)phenyl]-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
2-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyrazine
4-(oxolan-3-yl)-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-1,2,3-triazole
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
N-ethyl-5-[4-(oxolane-2-carbonyl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
4-[2-(4-fluorophenyl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(3-fluorophenyl)ethyl]piperidine-3-carboxamide
5-ethyl-N-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-(2-methyl-6-propylpyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
(1S,6R)-9-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(2,4-difluorophenyl)-3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
2-(5-acetylthiophen-3-yl)-N-[1-(thian-4-yl)piperidin-4-yl]acetamide
3-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
2-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-{[3-(difluoromethoxy)phenyl]methyl}piperidin-2-one
ethyl 1-{6-methylpyrazolo[1,5-a]pyrimidine-3-amido}cyclobutane-1-carboxylate
4-{2-[(3-methoxyphenyl)methyl]morpholine-4-carbonyl}-N-methylpyridin-2-amine
1-{1-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]piperidin-4-yl}-2-phenylethan-1-ol
3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
N-methyl-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-methyl-3-(1H-pyrazol-1-yl)propanamide
N,N-dimethyl-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]azepan-4-amine
methyl 4-[4-(2-methyloxane-2-carbonyl)piperazin-1-yl]benzoate
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)butanamide
(2S,3S)-3-methyl-2-[(2-methyl-1-benzofuran-5-yl)formamido]pentanamide
7-(1,3-benzothiazol-2-yl)-4-(prop-2-en-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
5-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamide
1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidin-3-ol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
1-(cyclohexylmethyl)-N-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-3-amine