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N-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N-methyl-1-(2-phenylethyl)piperidin-3-amine
(3R,4R)-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-ethylpiperidine-3,4-diol
(3S,4R)-3-benzyl-4-methyl-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-ol
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4-hydroxy-2-methylpyrimidine-5-carboxamide
1-({4-[(5-cyano-1,3-thiazol-2-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
5-[(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)methyl]-N,N-dimethylfuran-2-carboxamide
dimethyl[(5-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}thiophen-3-yl)methyl]amine
8-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-4-(4-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenyl)butan-2-ol
N-[(3-methoxyphenyl)methyl]-1-methyl-N-(2-methylpropyl)-1H-imidazole-5-carboxamide
6-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[7-oxo-5-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]cyclobutanecarboxamide
1-(2,3-dimethylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
(4aS,7aR)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-N-(1,2,4-thiadiazol-5-yl)benzamide
2-({2-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-(oxolane-2-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-[4-({[2-(1,3-benzothiazol-2-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-4-methylthiophene-2-sulfonamide
5-methyl-1-(3-methylphenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperazin-2-one
1-(cyclohexylmethyl)-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(2-hydroxyethyl)-9-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-4-cyclopropyl-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-3-carboxylic acid
3-(1-butyl-1H-pyrazol-5-yl)-1-[1-(thiophen-2-yl)propyl]urea
(1R,7S)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(2R,3R)-3-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-2-yl}pyridine
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidin-3-yl]acetamide
1-(2-ethoxyethyl)-N-[(5-methylfuran-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[5-(4-benzylpiperidin-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
5-(oxan-4-yl)-3-[3-(trifluoromethoxy)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
dimethyl[2-(3-{3-[4-(trifluoromethyl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)ethyl]amine
4-[(5-methylfuran-2-yl)methyl]-3-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)piperazin-2-one
N-(2-fluoro-4-methylphenyl)-2-{[1-(pyrrolidin-1-yl)cyclopentyl]formamido}acetamide
(3aR,6aR)-2-(2-methylfuran-3-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[N-(4-methylphenyl)methanesulfonamido]acetamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[(2-fluorophenyl)methyl]-3-{1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}propanamide
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3-propoxypiperidine
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-3-methylbutyl)-N-methylacetamide
1-[5-(6-methoxy-2H-chromen-3-yl)-4-phenyl-1H-imidazol-1-yl]propan-2-ol
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2E)-2-methylbut-2-en-1-yl](2-methylpropyl)amine
(1R,5R)-3-(5-fluoro-2-methylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-fluoroethyl)-5-methylpiperidin-2-one
6-{[(3R,4S)-1-(oxane-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
1-methyl-4-(5-methyl-1,3,4-oxadiazol-2-yl)-2-phenylpiperazine
(3aS,6aR)-5-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine