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N-cyclopropyl-5-[5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-ethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
(2S,4R)-1-(4-carboxybenzenesulfonyl)-4-(dimethylamino)pyrrolidine-2-carboxylic acid
2-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}benzoic acid
3-[4-(3-ethoxypropanoyl)-2-oxopiperazin-1-yl]benzonitrile
1-(2-methoxyethyl)-3-(4H-1,2,4-triazol-4-ylmethyl)piperidine
N-[(2-chlorophenyl)methyl]-4-methoxy-N-(propan-2-yl)cyclohexane-1-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidine
2-[(4-cyclopentylpyrimidin-2-yl)amino]-N-cyclopropylacetamide
(3S,4S)-4-cyclopropyl-1-(3-fluoropyridin-4-yl)pyrrolidine-3-carboxylic acid
N,6-dimethyl-4-oxo-N-[(4-phenoxyphenyl)methyl]-1,4-dihydropyridine-3-carboxamide
1-(ethanesulfonyl)-3,3-diphenylpiperidine
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
4-(4-{[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
ethyl 4-[(3-methoxyphenyl)methyl]-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxylate
{1-[3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propyl]piperidin-3-yl}methanol
N-[(3S,4R)-4-(4-methylphenyl)-1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]acetamide
4-(5-propylpyrimidin-4-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-(dimethylamino)-7-[3-(4-methoxyphenyl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(3-ethyl-1H-pyrazol-5-yl)pyridine-3-carbonitrile
3-({2-[(2S,4R)-4-amino-2-(methylcarbamoyl)pyrrolidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
(1S,5R)-3-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-methyl-5-{4-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[(2,3-difluorophenyl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
7-(1,3-benzothiazol-2-yl)-4-[(4-methoxy-3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(ethanesulfonyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(1-ethylpiperidin-4-yl)piperidine-3-carboxylate
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-(naphthalen-1-ylmethyl)-3-(1-propyl-1H-1,2,3,4-tetrazol-5-yl)urea
2-methyl-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}oxolane-2-carboxamide
8-[6-(dimethylamino)pyrimidin-4-yl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{5-[1-(3-methylphenyl)piperidin-4-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
5-{[1-(3-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
N-[(5-{[4-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
methyl (2S)-2-{3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}-3-phenylpropanoate
N-({1-[(3-ethenylphenyl)methyl]piperidin-3-yl}methyl)propane-2-sulfonamide
N-ethyl-N-(2-hydroxyethyl)-4-{[(4-methylphenyl)methyl]amino}benzamide
1-({5-[3-(1H-pyrrol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)piperidin-3-ol
6-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
(4aR,7aS)-1-(2-methoxyethyl)-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(2E)-3-phenylprop-2-en-1-yl]amine
N-{[3-methyl-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
ethyl 2-[(4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}piperidine-1-carbonyl)amino]acetate
{1-[(1,2-dimethyl-1H-indol-3-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol