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6-methyl-3-[4-(4-methylphenoxy)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
3-({3-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}methyl)-N-(pyridin-4-yl)benzamide
2-(pyrrolidin-3-yl)-N-[3-(4H-1,2,4-triazol-4-yl)phenyl]benzamide
2-(3,6-dimethylpyrazin-2-yl)-6-methyl-5-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-hydroxypropanamide
[3-(2-methoxyethyl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl]methanol
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}cycloheptanamine
1-methyl-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}acetamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1-(4-fluorophenyl)cyclopropane-1-carboxamide
6-chloro-2-(2-oxo-2-{spiro[azepane-4,2'-chromene]-1-yl}ethyl)-2,3-dihydropyridazin-3-one
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl]methylamine
N-benzyl-N-methyl-1-[2-(trifluoromethyl)benzoyl]piperidin-3-amine
2-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-5-methoxyphenol
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}furan-2-carboxamide
4-acetamido-N-ethyl-N-[2-(3-methylphenoxy)ethyl]benzamide
2-{4-[({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl}amino)methyl]phenoxy}ethan-1-ol
N-(3-chloro-4-methoxyphenyl)-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide
1-[(3-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(furan-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-[4-({3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]-1H-1,2,4-triazole
8-{[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]methyl}quinoline
{[(1R,5S,6S)-3-[(6-methoxy-2H-chromen-3-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
(1R,3S,5S)-8-{2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carbonyl}-8-azabicyclo[3.2.1]octan-3-ol
8-(2-aminoacetyl)-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-({2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2H-1,3-benzodioxol-5-ylmethyl)(2,3-dihydro-1-benzofuran-5-ylmethyl)(pyridin-3-ylmethyl)amine
3-(2-ethyl-1H-imidazol-1-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
1-(4-methoxyphenyl)-3-methyl-4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]piperazin-2-one
N-[1-(2-fluorophenyl)piperidin-4-yl]-2-(1H-pyrazol-1-yl)butanamide
6-(4-hydroxyphenyl)-2-[3-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-3-(1,2-oxazinan-2-yl)propan-1-one
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[3-(1,3-benzothiazol-2-yl)propyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-(2-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
(2S,4S)-N-methyl-1-(naphthalen-1-ylmethyl)-4-[(pyridin-3-ylmethyl)amino]pyrrolidine-2-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
(4aS,7aR)-4-[(2-methylphenyl)methyl]-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2S,4S)-4-amino-1-(4,5-dimethylthiophene-2-carbonyl)-N-methylpyrrolidine-2-carboxamide
1-(3-acetylphenyl)-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}urea
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazine
N-benzyl-N-methyl-2-(1-methylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(1S,6R)-9-(7-methanesulfonyl-4-methylquinazolin-2-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
2-ethoxy-6-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenol