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3-{1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidin-4-yl}-1,3-oxazolidin-2-one
1-({methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
(1S,6R)-9-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-3,9-diazabicyclo[4.2.1]nonane
N-(3,4-dimethoxyphenyl)-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
(4-{thieno[2,3-d]pyrimidin-4-yl}-1,4-oxazepan-6-yl)methanol
7-(1,3-benzothiazol-2-yl)-4-[(2,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)[(4-methyl-1,3-benzoxazol-2-yl)methyl]amine
3-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-1,3-oxazolidin-2-one
N-ethyl-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2,6-difluorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(pyrrolidin-3-yl)benzamide
3-(oxolan-3-yl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,2,4-oxadiazole
6-{2-[1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
2-{1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]pyrrolidin-3-yl}benzoic acid
(2S)-2-amino-2-cyclopropyl-1-(3,3-diphenylpiperidin-1-yl)ethan-1-one
N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]furan-3-carboxamide
6-[2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-2-methylpyrimidin-4-ol
methyl 3-[3-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)propanamido]thiophene-2-carboxylate
1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-(diphenylmethyl)-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
6-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
2-methoxy-4-[3-(pyridin-4-yl)azetidin-1-yl]pyridine-3-carbonitrile
11-{[(2,3-difluorophenyl)methyl]amino}-4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-methoxy-3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-(3-{[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]methyl}phenoxy)acetamide
4-(benzyloxy)-1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
(3aR,6aR)-2-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2H-1,3-benzodioxol-5-ylmethyl)-8-fluoro-3,4-dihydroquinazolin-4-one
N'-cyclooctyl-N-(2,3-dihydroxypropyl)-N-methylbutanediamide
methyl 2-(azepane-1-sulfonyl)-6-(pyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{3-[(3-methoxypyrrolidin-1-yl)sulfonyl]benzoyl}thiomorpholine
1-(4-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
{2-[2-amino-6-(thiophen-2-ylsulfanyl)pyrimidin-4-yl]phenyl}methanol
2-(cyclopent-1-ene-1-carbonyl)-1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)oxolane-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-phenoxyacetamide
N-(3-methoxyphenyl)-3-{[(2-methoxyphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
{3-[(2,4-difluorophenyl)methyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methanol
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-1H-1,2,4-triazole-5-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methoxyethan-1-one
N-(5-chloro-2-methoxyphenyl)-4-(6-oxo-1,6-dihydropyrimidin-4-yl)piperidine-1-carboxamide
5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyridin-2-amine
1-(3-{[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
1-(2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
5-(3-fluorophenoxymethyl)-N-(2-phenylpropyl)-1H-pyrazole-3-carboxamide
2-(dimethylamino)-N-[(4-hydroxyphenyl)methyl]-2-(2-methylphenyl)acetamide
4-methyl-6-(4-{[(3-propyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-amine
(2S)-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
1-{1-[(3-carbamoyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-3-carboxamide