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1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(2S)-2-({5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}formamido)-3-phenylpropanamide
(2S,4R)-4-amino-1-(3-cyclopentylpropanoyl)-N-methylpyrrolidine-2-carboxamide
2-(2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[(1-ethylpyrrolidin-2-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1-benzothiophene-2-carboxamide
2-cyclopentyl-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-phenylacetamide
1-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,4R)-4-(azepan-1-yl)-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
3-({4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
7-[3-(5-methylfuran-2-yl)butyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
methyl 3-[4-(1H-indole-2-carbonyl)-6-[(3-methoxyphenyl)methoxy]-2-oxo-1,4-diazepan-1-yl]propanoate
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
7-fluoro-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}quinazolin-4-amine
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-5-methyl-1H-indazole
1-(1-benzoxepine-4-carbonyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
1-methyl-2-[2-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-1H-1,3-benzodiazole
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}cyclobutanecarboxamide
N-[1-(4-phenylphenyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl)butan-2-ol
[(1-phenylcyclohexyl)methyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
5-chloro-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]pyrimidine
5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
2-(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}azetidin-3-yl)-1H-1,3-benzodiazole
methyl 5-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-7-thia-2-azatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene-3-carboxylate
6-(4-propylpiperazin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-{4-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-6-methylpyrimidin-2-yl}phenol
(4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1,4-oxazepan-6-yl)methanol
2-benzyl-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
3-{1-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperidin-4-yl}benzonitrile
7-[(2S)-2-phenylbutanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-(cyclopropylmethyl)-8-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-(2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidin-4-yl)piperidin-4-ol
2-(dimethylamino)-2-(2-methylphenyl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}acetamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(1H-indazol-1-yl)ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
(1R,2S,6R,7S)-N-(2-methylphenyl)-4-azatricyclo[5.2.2.02,6]undecane-4-carboxamide
4-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}-1λ6-thiomorpholine-1,1-dione
14-ethyl-6-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(4aR,8aS)-N,N-dimethyl-1-[(2E)-2-methylbut-2-enoyl]-decahydro-1,6-naphthyridine-6-sulfonamide
1-[(3-fluorophenyl)methyl]-4-[2-(phenylsulfanyl)acetyl]piperazin-2-one
1-{4-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]piperidin-1-yl}ethan-1-one
N4,N4,N6-trimethyl-N6-[2-(2-methylpiperidin-1-yl)ethyl]pyrimidine-4,6-diamine
2-methyl-6-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}pyrimidin-4-ol
6-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoxaline
2-ethyl-1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)butan-1-one
N4-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-6-methylpyrimidine-2,4-diamine
(2R,3R)-3-{[3-(1H-indazol-1-yl)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol