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N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
3-methyl-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1-phenyl-1H-pyrazol-5-amine
1-cyclopentyl-4-[3-(piperidin-3-yl)benzoyl]piperazine
4-(5-chloro-2-methoxypyridin-4-yl)-6-(morpholin-4-yl)pyrimidin-2-amine
ethyl 5-(5-ethyl-1,2-oxazole-3-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(2-methoxyphenyl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
2-(3-chloro-4-hydroxyphenyl)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}acetamide
2-(4-fluoro-3-methylphenyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-{5-methyl-2-oxo-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperazin-1-yl}benzonitrile
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(4-ethylpiperazin-1-yl)acetamide
1-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-methyl-3-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)quinoxaline
2-[4-(hydroxymethyl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(5-oxo-1-propylpyrrolidin-3-yl)acetamide
N3-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-1,3-dicarboxamide
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-fluorophenyl)ethan-1-one
7-cyclohexyl-2-(1-methyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,2,5,6-tetramethylpyrimidin-4-amine
2-[(isoquinolin-5-yloxy)methyl]-N-(1-propylcyclopropyl)-1,3-oxazole-4-carboxamide
3-{1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-(6-methoxypyridine-3-carbonyl)-4-methylpiperidine-3,4-diol
4-{1-[6-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl}benzoic acid
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
(1R,5S,8S)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
1-[4-(morpholin-4-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N'-(3-chloro-4-fluorophenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanediamide
4-[3-(4-benzylpiperidine-1-carbonyl)piperidin-1-yl]-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-({2-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
methyl 4-methoxy-3-({[2-(N-methylmethanesulfonamido)ethyl]carbamoyl}amino)benzoate
N-(3-oxo-3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propyl)acetamide
3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-N-(1,2,3-thiadiazol-5-yl)benzamide
N-cyclopropyl-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridine-4-carboxamide
ethyl 2-[2-(5-{[3-(1H-imidazol-1-yl)propyl]carbamoyl}thiophen-2-yl)pyrrolidin-1-yl]acetate
(3R,9aR)-3-benzyl-8-(4-fluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{4-[(4-ethyl-3,3-dimethylpiperazin-1-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
(3S,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-methyl-2-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-indole
1-(4-fluorophenyl)-4-(piperidin-3-ylmethyl)-1,4-diazepane
2,2-diethyl-4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}morpholine
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(methoxymethyl)-3-methyl-1H-pyrazole
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}urea
(1S,5R)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S)-N-(4-acetylphenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
8-(5-methylthiophene-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one