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N-[2-(dimethylamino)ethyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-{7-[(6-ethoxypyridin-3-yl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methylpropan-1-one
3-(1H-imidazol-1-ylmethyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
4-[4-(piperidin-3-yl)benzoyl]thiomorpholine
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-5-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[3-(trifluoromethyl)piperidin-1-yl]pyrimidine
5-(2,4-difluorophenoxymethyl)-N,N-dipropyl-1,2-oxazole-3-carboxamide
ethyl 2-(4-{2-methylthieno[2,3-d]pyrimidin-4-yl}morpholin-3-yl)acetate
2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1,3-thiazole
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}quinoline
N-[(3S,4R)-1-(6-cyclopropylpyrimidin-4-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-benzyl-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazin-2-one
8-chloro-2-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}quinolin-4-ol
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
2-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}-3,5-dimethoxybenzoic acid
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
N-[(2-methoxyphenyl)methyl]-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(3S,4R)-4-(3-fluorophenyl)-1-(2-methoxy-5-methylbenzoyl)pyrrolidine-3-carboxylic acid
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)(1,2-oxazol-3-ylmethyl)amine
N,N-dimethyl-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
8-(5-chloropyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(3-hydroxyphenyl)methyl]-N-methylacetamide
(2-{[4-(1-ethylpyrrolidine-3-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
N-cyclohexyl-8-fluoro-N-[(1-methyl-1H-pyrazol-4-yl)methyl]quinoline-2-carboxamide
3-methyl-7-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidine-3-carboxamide
4-methoxy-6-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-2-amine
1-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-phenylpyrrolidine-3-carboxylic acid
4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-2-(pyrrolidin-1-yl)benzamide
1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
6-(3-ethoxy-4-methoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
N-[(2-chlorophenyl)methyl]-3-[1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperidin-3-yl]propanamide
5-({3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
4-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-ethylpiperazin-2-one
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-(furan-2-yl)propan-1-one
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-ethoxy-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
8-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
2-(pyridin-3-yl)-7-(thiophene-2-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-(azetidine-1-carbonyl)-N-[(3-methylphenyl)methyl]-1-propyl-1H-1,3-benzodiazol-2-amine
4-methyl-2-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,3-thiazole
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-6-ethyl-N,1,5-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(3-acetylphenyl)-1-methyl-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-(1H-indol-1-ylmethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-(2-oxo-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one