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1-(5-ethylthiophene-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
5,7-dimethyl-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}pyrazolo[1,5-a]pyrimidine
1-(2-ethylbutanoyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-[(3S,4R)-4-propyl-1-(pyrazin-2-yl)pyrrolidin-3-yl]acetamide
5-methyl-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)thiophene-2-carboxamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2,6-dimethylpyridine-4-carboxamide
1-(1-carbamoylethyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
2-tert-butyl-5-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]pyrimidin-4-ol
6-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)aniline
methyl (2S,4R)-1-methyl-4-[2-(pyridin-4-ylsulfanyl)acetamido]pyrrolidine-2-carboxylate
1-(2-cyclopropyl-4-hydroxypyrimidine-5-carbonyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}ethan-1-one
8-(2,3-dihydro-1-benzofuran-5-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,4R)-N,N-diethyl-1-methyl-4-[2-methyl-5-(propan-2-yl)furan-3-amido]pyrrolidine-2-carboxamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)morpholine-4-carboxamide
8-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-(6-methoxypyridin-3-yl)pyridine-3-carboxamide
2-(oxolan-2-ylmethyl)-9-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(3S,4S)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
(1R,5S,6S)-6-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
1-methyl-4-{[4-(methylsulfamoyl)phenyl]methyl}piperazine-2-carboxylic acid
N2,N2,N4,N4-tetramethyl-7-(1-propyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(3aR,6aR)-2-[(4-fluoro-3-methylphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-5-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-6-methyl-3,4-dihydropyrimidin-4-one
8-[5-chloro-2-(methylamino)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(5-methyl-2-phenylfuran-3-carbonyl)pyrrolidin-3-yl]methanol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-9H-purin-6-amine
(4S,4aS,8aS)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
2-(dimethylamino)-2-(4-methylphenyl)-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}acetamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole
N-[cyclopropyl(pyridin-2-yl)methyl]-3-[(4-fluorophenyl)formamido]-N-methylpropanamide
N-{[4-hydroxy-1-(thiophene-2-carbonyl)azepan-4-yl]methyl}morpholine-4-carboxamide
5-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
1-methyl-N-[2-(propan-2-yloxy)ethyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
2-[3-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)phenoxymethyl]pyridine
2-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrazine
2-[4-(6-cyanopyridine-3-carbonyl)morpholin-3-yl]-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}acetamide
3-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyridin-4-yl)propanamide
4-(4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl)piperidin-4-ol
2-[2-(8-fluoroquinoline-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetic acid
3-(hydroxymethyl)-1-(5-methylthiophene-2-carbonyl)piperidin-3-ol
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-fluoropyridine
{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}({[4-(1H-pyrazol-1-yl)phenyl]methyl})amine
1-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}cyclopropane-1-carboxamide
4-[4-({[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]-2-methylbut-3-yn-2-ol