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2-(dimethyl-1,2-oxazol-4-yl)-2-{[(8-methoxyquinolin-5-yl)methyl](methyl)amino}acetic acid
2-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyridin-2-yl)ethan-1-ol
N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
N-[3-(furan-2-yl)phenyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
3-[(4-fluorophenyl)formamido]-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}oxy)benzamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-(3-methoxypropyl)piperidine
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
(1R,5R)-3-methanesulfonyl-6-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(4aR,7aS)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-{4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-(furan-2-ylmethyl)acetamide
1-[3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenyl]ethan-1-one
5-[2-(4-fluorophenyl)morpholine-4-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
ethyl 1-(thiophene-3-sulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
(3S,4R)-4-(3-fluorophenyl)-1-[1-(4-fluorophenyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(thiophen-2-ylmethyl)piperidine
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-[(2R)-2-methylpyrrolidine-2-carbonyl]piperazine
2-(2-{5-[(5-ethylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrrol-1-yl)pyrimidine
3-(2-methoxyphenyl)-4-(3-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(pyridine-4-carbonyl)piperidine-3-carboxylate
1-[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)benzoyl]piperidine
5-(2-chloro-4-methoxyphenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
1-{5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}ethan-1-one
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-N-(5-methylpyridin-2-yl)acetamide
N-{2-[({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]ethyl}acetamide
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(thian-4-yl)piperazine
methyl 3-({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}carbamoyl)propanoate
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
N-cyclopropyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-(thiophen-3-ylmethyl)acetamide
8-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}phenyl)acetamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
5-oxo-1-[4-(propan-2-yl)phenyl]-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
2-[2-(3-chlorophenyl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide
5-(5-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}furan-2-yl)-1H-pyrazole
2-(2-chloro-4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
2-{1-[4-(1H-1,2,4-triazol-1-yl)butyl]piperidin-3-yl}propan-2-ol
2-methyl-N-{2-[methyl(phenyl)amino]propyl}imidazo[1,2-a]pyrimidine-3-carboxamide
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[(4aS,8aR)-4a-(hydroxymethyl)-6-[(3-methylthiophen-2-yl)methyl]-decahydro-1,6-naphthyridin-1-yl]acetamide
7-[4-(1H-pyrazol-5-yl)phenyl]-1,2,3,4-tetrahydroisoquinoline
4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
N-[(1R)-2-hydroxy-1-phenylethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide