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1-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
(3aS,6aS)-2-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-methoxyethan-1-one
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]propanamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}propane-1-sulfonamide
1-[(2,4-dimethylphenyl)methyl]-4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
1-{2-[4-(2-phenoxyethyl)piperazin-1-yl]pyrimidin-4-yl}piperidin-4-ol
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
5-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1,3-thiazol-2-amine
3-[(3-fluorophenyl)methyl]-N-methyl-N-(thiophen-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[4-(2-ethoxypyridine-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
N-({1-[(3-cyanophenyl)methyl]piperidin-3-yl}methyl)cyclohexanecarboxamide
4-amino-N-[2-(2-phenoxyethoxy)phenyl]pyridine-2-carboxamide
N-({1-[(4-chlorophenyl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
5-{3-[4-(2-chlorophenoxy)piperidin-1-yl]-3-oxopropyl}-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
2-(cyclopropylmethyl)-8-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-ethoxy-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)furan-2-carboxamide
2-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]ethoxy}ethan-1-ol
8-fluoro-N-[(4-methanesulfonylmorpholin-2-yl)methyl]quinoline-2-carboxamide
4-(1-ethylpiperidin-4-yl)-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-{1'-[(1-methyl-1H-indol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-(5-acetamido-2-fluorophenyl)-4-(thian-4-yl)piperazine-1-carboxamide
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[4-(propylsulfamoyl)phenyl]urea
5-(azepane-1-carbonyl)-N-methyl-1-(2-methylpropyl)-4-oxo-N-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
2-(adamantan-1-yl)-N-(3-ethoxypropyl)-4-hydroxypyrimidine-5-carboxamide
7-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[1'-(3,5-difluoropyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-methoxy-2-{[methyl({[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenol
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-methoxyacetamide
[(5-fluoro-1H-indol-2-yl)methyl]({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
2-{3-[1-(but-2-yn-1-yl)-1H-pyrazol-3-yl]phenyl}-3-fluoropyridine
N-(2,3-dihydro-1H-inden-2-yl)-2,4-difluoro-3-methoxy-N-methylbenzamide
6-(furan-3-yl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
2-[5-(5-acetylthiophen-2-yl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-(1-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
2-(3-{[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]methyl}phenoxy)acetamide
N,N,4-trimethyl-3-({methyl[2-(pyrrolidin-1-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[(1S,5R)-3-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
(3S,4S)-4-(piperidin-1-yl)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
4-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(cyclopentylmethyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
2-[3-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]ethan-1-amine
5-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N4-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]-5-ethylpyrimidine-2,4-diamine
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
4-chloro-N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1-methyl-1H-pyrazole-3-carboxamide
4-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)-2,6-dimethoxyphenol