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8-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
5-[1-(benzenesulfonyl)cyclopropyl]-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
2-(2-hydroxyethyl)-8-[2-(3-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-phenylurea
6-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(oxan-4-yl)piperidine-3-carboxamide
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(methyl)(quinolin-8-ylmethyl)amine
1-[(3-{[1-(naphthalene-2-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
2,6-dimethyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-4-carboxamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
2-chloro-6-methoxy-4-[1-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-imidazol-2-yl]phenol
5-tert-butyl-N-[3-(propan-2-yloxy)propyl]-1,3,4-oxadiazol-2-amine
2-(4-fluoro-2-methoxyphenyl)-1,3-benzothiazole
(1S,4S)-2-(2-chlorophenyl)-5-[(3-methylquinoxalin-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-ethyl-2-[2-(trifluoromethoxy)phenyl]pyridine-4-carboxamide
1-(4-tert-butylbenzoyl)-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
9-(3-methoxybenzoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1,3-dimethylpiperazin-2-one
8-methoxy-5-[6-(morpholine-4-carbonyl)pyrazin-2-yl]quinoline
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
(1S,6R)-9-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(2-methylbutanoyl)-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3,3-dimethyl-1-[(5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyrimidin-4-ylmethyl)pyridin-2-amine
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-[(1-methylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-3-carboxylate
2,5-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(2,5-dioxoimidazolidin-1-yl)-N-(1-ethylpiperidin-4-yl)-N-[2-(pyridin-2-yl)ethyl]acetamide
1-(1-methyl-1H-pyrazol-4-yl)-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
N-[(4-phenyloxan-4-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-methyl-1-(3-methylbutyl)-4-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N4-methyl-N4-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1,3,6-trimethyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
N'-{[1-(9H-fluoren-2-ylmethyl)pyrrolidin-3-yl]methyl}ethanediamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl]methanol
1-[4-({3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
3-{[4-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
2-butoxy-1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-{4-[3-(1H-pyrazol-1-yl)phenyl]phenyl}ethan-1-ol
(3S,9aR)-8-[(2-methoxyphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(3-methoxyphenyl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}furan-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-propyl-1,2-oxazole-3-carboxamide
7-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-(4-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
4-(1-{1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
4-chloro-N-ethyl-1-methyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-1H-pyrazole-3-carboxamide
dimethyl({[4-methyl-5-(1-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine