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2-{4-[4-ethoxy-3-(hydroxymethyl)phenyl]-1H-1,2,3-triazol-1-yl}-N-methylpropanamide
1-[3-(dimethylamino)pyrazin-2-yl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-ethyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)propanamide
1-{[4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]methyl}piperidine
4-[2-(1H-imidazol-1-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
N-(butan-2-yl)-3-(1,2-oxazinan-2-yl)-N-(pyridin-4-ylmethyl)propanamide
(3R,4S)-1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-propylpyrrolidin-3-amine
1-cyclopentyl-4-[4-methoxy-2-(4-methoxypiperidine-1-carbonyl)phenoxy]piperidine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopent-1-ene-1-carboxamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(5-methylthiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-(4-methylphenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-[1-(2-amino-6-methylpyrimidine-4-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[3-(4-fluorophenoxymethyl)-1-propyl-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
1-[(2,3-difluoro-4-methylphenyl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-[3-(4-chlorophenyl)-4-methyl-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
5-({2-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1-methyl-1H-1,2,3,4-tetrazole
1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
2-{5-[4-(2-fluorophenyl)piperazin-1-yl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-2-methyl-4-phenylpyridine-3-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,3-dihydro-1H-inden-1-yl)-1H-pyrazole-3-carboxamide
({4-ethyl-5-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-[({[3-(2-{4-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
N-methyl-N-(4-methyl-1-phenylpentyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
2-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-N-methylacetamide
2-ethyl-5-{2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydropyrimidin-4-one
3-(azetidine-1-sulfonyl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]propanamide
2-butyl-8-[2-(2-methoxyethoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3,5-dimethyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]adamantane-1-carboxamide
N-[2-(dimethylamino)ethyl]-1-[1-(2-ethylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
4-(5-fluoro-2-methoxyphenyl)-1-methyl-1H-pyrazol-5-amine
N-(3-methoxypropyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-ylmethyl)acetamide
(4aR,8aS)-1-{[4-(trifluoromethyl)phenyl]methyl}-6-[2-(3,4,5-trimethoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-2-one
5-[(1-benzothiophen-2-ylmethyl)amino]-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(4-methoxyphenyl)butanamide
N-{2-[1-cyclohexyl-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N,7,8-trimethyl-2-(1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
3-[(4aR,7aS)-4-(3-fluorobenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-(pyrrolidin-1-ylmethyl)-1-(quinoline-3-carbonyl)piperidin-3-ol
1-[6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrimidin-4-yl]piperidin-4-ol
2-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)benzonitrile
5-chloro-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-1H-indole-2-carboxamide
(2S,4S,5R)-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-(2,4-dichlorophenoxy)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}acetamide
N-cyclopentyl-1-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
3-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]sulfonyl}-N-(prop-2-en-1-yl)benzamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})amine