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N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
1-{[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
N-[(2R)-1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-oxobutan-2-yl]acetamide
methyl 4-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]benzoate
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-methyl-4-{3-[4-(3-methylphenyl)piperazine-1-carbonyl]phenyl}butan-2-ol
1-[(3-methoxyphenyl)methyl]-4-(3-methoxypyrazin-2-yl)piperazin-2-one
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-butyl-4-(2-methoxypyridine-4-carbonyl)-1-methylpiperazin-2-one
5-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-1-propylpiperidin-2-one
3-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-4-(furan-3-ylmethyl)piperazin-2-one
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-hydroxyethan-1-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-methyl-2-phenylpropanamide
3-(4-chlorophenyl)-4-(1-ethyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]azocane-1-carboxamide
2-cyclopropyl-8-[(2-fluoro-5-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(cyclopropylmethyl)-8-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-N-[(2-fluorophenyl)methyl]propanamide
1-(2-cyclohexylethyl)-3-({[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-methoxy-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[2-(pyridin-2-yl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
2-(2-acetylbenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
benzyl[(4-methyl-1H-imidazol-5-yl)methyl](1,3-thiazol-2-ylmethyl)amine
3-(2-methanesulfonylethyl)-1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
6-{[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylacetamide
2-{methyl[3-(oxolan-2-yl)propyl]amino}acetic acid
2-(3-{1-[2-(diethylamino)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine-4-carbonitrile
2-(3-{[3-(3-methylphenyl)piperidin-1-yl]methyl}phenoxy)acetamide
1-{3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}propan-1-one
methyl 7-oxo-3-(oxolane-2-carbonyl)-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{5-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(pyrazin-2-ylmethyl)amine
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
N-(3-methoxyphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
3-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanoic acid
3-(piperazine-1-carbonyl)-N-[3-(1H-pyrazol-1-yl)propyl]benzene-1-sulfonamide
5-acetyl-N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
1-(azepan-1-yl)-3-[3-({[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
methyl 5-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
7-(propan-2-yl)-2-[4-(1H-pyrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-(9H-purin-6-yl)piperidin-4-amine
3-methyl-8-{[4-(2-phenylethoxy)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one