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(3aR,6aR)-2-[(4-tert-butylphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4S)-4-phenyl-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-oxazolidin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(2S,4R)-4-amino-1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(3-methylbutyl)-1,2-oxazole-3-carboxamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
N-[2-(2-fluorophenyl)-1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
4-(4-methylpiperazine-1-carbonyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridin-2-amine
3-(piperidin-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
4-(2-methoxyphenoxy)-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
3-{1-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-1H-imidazol-2-yl}phenol
(1S,5R)-3-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
(4aR,7aS)-1-(2-methylpropyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-1-one
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-phenyl-1,2-oxazole-5-carboxamide
methyl (2R,4S)-1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4-hydroxypiperidine-2-carboxylate
(2R,6S)-4-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2,6-dimethylmorpholine
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
4-(1-butyl-1H-imidazol-2-yl)-1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidine
2,8-dimethyl-4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]quinoline
2-(1-methylpiperidin-4-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}oxane-2-carboxamide
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
8-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-cyclopentyl-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-(4-methoxy-2-methylphenyl)-N-methylpyridine-3-carboxamide
2-(3,4-dichlorophenyl)-4-[1-(pyrimidin-2-yl)piperidin-4-yl]morpholine
[(2S,6S)-4-cyclohexyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-{1-[2-(4-fluorophenyl)azetidin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1,2,3-thiadiazole-4-carboxamide
(3S,4S)-1-(5-methoxypyrimidin-2-yl)-4-propylpyrrolidine-3-carboxylic acid
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(pyridin-2-yl)propan-1-one
6-oxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-(methoxymethyl)pyrimidin-4-amine
3-(furan-2-ylmethyl)-1-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}urea
3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-[(2S)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(4-fluorophenyl)ethyl]-2-(2-oxopiperidin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
2-(2-methylpropyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(dimethylamino)ethyl]-5-(3-hydroxy-2-methylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
2-(4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperazin-1-yl)pyrazine
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]propanamide
N-{1-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[1-(1H-indol-5-yl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(2-fluorophenyl)methyl]-5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-[(3R,5S)-5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]pyrrolidin-3-yl]-2-phenoxyacetamide
ethyl 2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]acetate