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2-methanesulfonyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]acetamide
(2E)-N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-[(2,5-difluorophenyl)methyl]-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3-propyl-1H-pyrazole-4-carboxamide
7-fluoro-4-methyl-2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
ethyl 1-(cyclopropylmethyl)-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
N-ethyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(pyridin-4-ylmethyl)acetamide
N-methyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
2-amino-8-(2-ethylphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
N-({7-[5-(4-methoxyphenyl)furan-2-carbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-methylpyrazine-2-carboxamide
1-(2-methoxyethyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-(2,5-dimethylphenyl)-3-{[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}propanamide
1-(1-methylpiperidin-4-yl)-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
2-[4-({4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazin-1-yl]pyrimidine
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(1H-1,2,4-triazol-1-yl)propanamide
6-(benzyloxy)-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
({5-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-2-methoxyphenyl}methyl)dimethylamine
2-[4-fluoro-2-(trifluoromethyl)phenyl]-5-(methanesulfonylmethyl)pyridine
5-(dimethoxy-1,3,5-triazin-2-yl)-8-methoxyquinoline
4-(methylsulfanyl)-2-[(2-oxo-6-phenyl-1,2-dihydropyridin-3-yl)formamido]butanoic acid
1-{3-[4-(5-tert-butyl-1H-pyrazol-3-yl)-1H-1,2,3-triazol-1-yl]propyl}pyrrolidin-2-one
1-{1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carbonyl}-N,N-diethylpiperidine-3-carboxamide
1-(1-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(propan-2-yl)-1H-imidazole
2-[methyl(pyridin-4-ylmethyl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
methyl N-(1-oxo-1-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}propan-2-yl)carbamate
2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1,2-dihydrophthalazin-1-one
1-(azocan-1-yl)-3-(5-{[bis(prop-2-en-1-yl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]benzamide
6-({4-[3-(dimethylamino)-2-hydroxypropoxy]phenyl}methyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[2-(1H-indol-1-yl)ethyl]-N,1,5,6-tetramethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{2-[(4-chlorophenyl)methyl]-1,3-benzoxazole-5-carbonyl}-1,4-oxazepan-6-ol
4-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-6-methylquinoline
2-acetamido-N-[3-(3-ethylphenoxy)propyl]-N,3-dimethylbutanamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-5-cyclopropyl-1,3-oxazole-4-carboxamide
2-(2-methylpropyl)-N-(1,2,3-thiadiazol-5-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
3-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
N-[2-(methylsulfanyl)ethyl]-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
4-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-4-{1H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
2-(3-ethoxyphenyl)pyridine-3-carboxamide
3-{1-[3-(furan-2-yl)propanoyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
5-ethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine