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3-{4-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]phenyl}prop-2-yn-1-ol
(1R,2S)-N-butyl-2-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclohexane-1-carboxamide
1-(2-fluorophenyl)-4-{4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}piperidin-4-ol
2-{1-ethyl-2,4-dioxo-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
5-(methoxymethyl)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-methyl-3-phenylpiperazin-1-yl)-2-(pyrrolidin-1-yl)ethan-1-one
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(1H-imidazol-2-yl)benzoyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-1-(4-methylphenyl)piperazin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-N-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
5-(thiomorpholine-4-carbonyl)-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-1-(3,5-dimethylphenyl)piperazin-2-one
2-{5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
N-(1,3-benzoxazol-2-ylmethyl)-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
(4aS,8aR)-6-(2-aminopyrimidin-4-yl)-1-[2-(2-hydroxyethoxy)ethyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}amino)methyl]phenol
1'-(2,1,3-benzothiadiazol-5-ylmethyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-cyclohexyl-5-[5-(methoxymethyl)furan-2-yl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-(dimethyl-1,2-oxazol-4-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
(1R,5S)-8-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
4-({1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1,5-dimethyl-1H-pyrazole
(2S,4R)-1-benzyl-N-methyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
N-benzyl-2-[4-(4-{[2-(3-phenylpyrrolidin-1-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
1-(cyclopropylmethyl)-5-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-methoxy-3-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)phenol
3-({1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
4-({1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]azetidin-3-yl}oxy)benzoic acid
N-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-{1-[(3-methoxyphenyl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
5-({2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
2-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
2-methyl-6-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3-dihydropyridazin-3-one
2-({[1-(2-benzyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
5-benzyl-3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
N-{5-[2-(2,3-dihydro-1H-isoindol-2-yl)acetamido]-2-methoxyphenyl}benzamide
2-(ethylamino)-4-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,3-thiazole-5-carboxamide
3-(4-{[5-(2-cyanophenyl)furan-2-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
(3S,4S)-1-{[2-(cyclopentyloxy)phenyl]methyl}-4-[(dimethylamino)methyl]piperidin-3-ol
1-methyl-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(1H-indazole-3-carbonyl)piperidin-4-yl]propanamide
4-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-N-methylpyridin-2-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[1-(methoxymethyl)cyclopropyl]-N-methylacetamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-methylpyrimidine-2,4-diamine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one