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1-{2-[4-(3-methylphenoxy)piperidine-1-carbonyl]phenyl}ethan-1-one
methyl 2-{7-chloro-3-[(cycloheptylamino)methyl]-2-oxo-1,2-dihydroquinolin-1-yl}acetate
1-cyclohexyl-3-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}urea
diphenyl[1-(pyrazine-2-carbonyl)piperidin-4-yl]methanol
2-(2,3-dimethoxyphenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
2-(azocane-1-carbonyl)-7-fluoro-3-methyl-1H-indole
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-(pyridin-3-ylmethyl)piperidin-4-yl]acetate
(1R,7S)-3-[2-(4-methylphenyl)ethyl]-6-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-(4-{3-[4-(3-methylphenyl)piperazin-1-yl]propanoyl}morpholin-3-yl)acetic acid
3-{[(1R,2R)-2-hydroxycyclohexyl]methyl}-3H,4H-pyrido[2,3-d]pyrimidin-4-one
N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carboxamide
N4-cyclopropyl-6-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyrimidine-2,4-diamine
3-{methyl[2-(trifluoromethyl)pyrimidin-4-yl]amino}-1-phenylpropan-1-ol
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-pyrazole-3-carboxamide
4-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]-1H-pyrrole-2-carbonitrile
N-{1-[(8-methoxyquinolin-2-yl)methyl]pyrrolidin-3-yl}acetamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-(2-cyclohexylethyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
ethyl 2-{1-[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-inden-2-yl]-N-methylformamido}acetate
4-{4-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}-2-methylbut-3-yn-2-ol
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
(3S,4S)-1-(1-benzoylpiperidin-4-yl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
1-[3-(2-methyl-1H-indol-1-yl)propanoyl]imidazolidin-4-one
2-(3-{[benzyl(methyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
(2S)-2-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}-3-phenylpropanoic acid
3-(morpholine-4-sulfonyl)-5-(quinolin-5-yl)benzoic acid
5-(oxolane-2-carbonyl)-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[3-(azocan-1-yl)-3-oxopropyl]-6-methyl-1,2-dihydropyridin-2-one
N-[(4-methyl-5-oxomorpholin-2-yl)methyl]-2-(thiophen-3-yl)acetamide
1-(2,6-dimethylpyridin-4-yl)-4-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperazine
2-{1-methyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}pyridine
2-(2,5-dimethoxyphenyl)-N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
2-methyl-8-[4-(trifluoromethyl)pyridin-2-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-{[5-(4,5-dimethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
2,6-dimethyl-5-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
2-(2-methoxyethyl)-9-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(morpholin-3-yl)acetamide
N-(6-chloro-2-methylpyridin-3-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-methyl-3-(2-phenylethyl)-8-propyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
2-{1'-[(3-fluoro-5-methylphenyl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
methyl 4-[2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetyl]piperazine-1-carboxylate
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]cyclopentanamine
N-methyl-N-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}oxan-4-amine
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[2-(pyridin-3-yl)ethyl]morpholine-2-carboxamide
3-(cyclopropylmethyl)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidine-3-carboxylic acid
3-chloro-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}pyridine