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1-(1H-imidazol-2-ylmethyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
(1S,4S)-2-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-3-(hydroxymethyl)piperidin-3-ol
(2S,4R)-1-benzyl-N-methyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-2-(2-methylphenyl)pyrimidine
4-methyl-6-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine
2-{8-[(3-hydroxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
1-[benzyl(methyl)amino]-3-(4-{[bis(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
methyl({[3-methyl-1-(2-{octahydropyrrolo[1,2-a]piperazin-2-yl}ethyl)-1H-pyrazol-4-yl]methyl})(prop-2-yn-1-yl)amine
2-benzyl-N-[2-(pyridin-3-yl)ethyl]-1,3-benzoxazole-5-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-methyl-3-[1-(oxane-4-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4'-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-cyclobutanecarbonyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-chloro-4-fluoro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}benzamide
3-fluoro-5-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]benzonitrile
1-methyl-3-(2-methylpropyl)-N-[2-(4-sulfamoylphenyl)ethyl]-1H-pyrazole-5-carboxamide
4-[(4-methoxyphenyl)methyl]-1-{[4-(methylsulfanyl)phenyl]methyl}-1,4-diazepan-5-one
7-[(2,3-difluorophenyl)methyl]-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decane
1-(carbamoylmethyl)-N-[(3-phenylphenyl)methyl]piperidine-3-carboxamide
5-methyl-3-(4-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)-1,2,4-oxadiazole
4-(1-{4-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}ethyl)morpholine
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[3-(4-methylphenyl)phenyl]piperidin-4-amine
5-methyl-3-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}-1H-indole-2-carboxylic acid
1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
ethyl 1-acetyl-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(3-methoxypropyl)-5-methyl-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}thiophene-2-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-5-methyl-N-(pyridin-3-ylmethyl)pyrazine-2-carboxamide
3,5-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,1-benzoxazole-3-carbonyl)piperidin-3-ol
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-(3-methoxyphenoxy)azetidine
4-[2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetyl]piperazin-2-one
5-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pentan-1-one
N-{1-[3-cyclopentyl-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
(1s,4s)-4-hydroxy-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]cyclohexane-1-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)acetamide
2-[(3,5-difluorophenyl)methyl]-8-(piperidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N,2-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]thiomorpholine
N-(3-hydroxyadamantan-1-yl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(3S,4R)-1-[2-(diethylamino)ethyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
8-{[2-(cyclopentyloxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(morpholin-4-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-3-yl)acetamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}propanamide
3-(2-hydroxyphenyl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
4-[3-(3-phenylpropanoyl)piperidine-1-carbonyl]benzonitrile
4-{[3-(3,6-dimethylpyrazin-2-yl)phenyl]methyl}morpholine
(3S,4S)-4-methyl-1-[2-(morpholin-4-yl)benzoyl]piperidine-3,4-diol