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4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-fluoro-3-methylphenyl)methyl]piperidine
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
2-[1-cyclopentyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methylacetamide
{2-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)oxy]ethyl}dimethylamine
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-(quinazolin-4-yloxy)ethan-1-one
N6-cyclopentyl-N5-methyl-N5-[(1-methyl-1H-pyrazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[5-(1-benzylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
8-(3-ethoxypropanoyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-ethyl-8-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{5-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
methyl 4-(3-{[(5-methylpyrazin-2-yl)methyl]amino}propanamido)benzoate
2-ethyl-6-methyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
2-{2-methylimidazo[1,2-a]pyridin-3-yl}-1-[4-(4-methylphenyl)piperazin-1-yl]ethan-1-one
N-[(3S,4R)-1-(2-hydroxyacetyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-(cyclohex-3-ene-1-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
(1S,3R)-N-(2,3-dihydro-1H-inden-4-yl)-3-[3-(methylsulfanyl)propanamido]cyclopentane-1-carboxamide
N,N,8-trimethyl-2-[2-(morpholin-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
N-cyclopentyl-4-[4-(3-methylphenoxy)piperidin-1-yl]-4-oxobutanamide
6-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methoxyacetamide
6-(azepan-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
5,6-dimethyl-1-(3-methylpyrazin-2-yl)-1H-1,3-benzodiazole
3-amino-1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]pyrrolidine-3-carboxylic acid
9-[(2-butyl-1H-imidazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N-({1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}methyl)cyclopropanecarboxamide
N-(propan-2-yl)-1-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(2-ethoxyphenyl)pyridine-4-carbonitrile
N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N-benzyl-N,1-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methoxy-5-{1-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(3-methyl-1,2-oxazol-5-yl)methyl]benzamide
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-methylpiperidine-3-carboxamide
8-{2-[(4-chlorophenyl)methyl]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
4-cyclobutyl-6-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidin-2-amine
N-{2-[4-(dimethylamino)phenyl]ethyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(piperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}phenoxy)acetic acid
N-[(4-fluorophenyl)methyl]-5-[(3-hydroxy-2,2-dimethylpropyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{2-[1-(3-hydroxypyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
3-{[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]methyl}-5-(propan-2-yl)-1,2,4-oxadiazole
2-ethyl-9-(2-methoxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-oxo-4-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]butanoate
5-chloro-6-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-2-methylpyrimidin-4-ol
N-cyclopentyl-3-{[3-(1H-1,2,4-triazol-1-yl)propyl]sulfamoyl}benzamide
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-(3-cyanopyridin-2-yl)-4-(3-phenylpropyl)piperidine-4-carboxylic acid