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4-(4-fluoro-3-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
3-(1-ethyl-1H-imidazol-2-yl)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine
1-(furan-2-ylmethyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]piperidine-3-carboxamide
2-(3-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-[(4-fluorophenyl)methyl]-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
N-(2-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-2-yl}ethyl)acetamide
N-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidine
1-cyclopropanecarbonyl-N-[3-(1H-indol-2-yl)phenyl]pyrrolidine-2-carboxamide
N-(3-hydroxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl)acetamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-4-carboxamide
methyl N-{2-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}carbamate
2-{4-[(6-chloroquinolin-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
[(3R,4R)-1-{[3-(cyclopentyloxy)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-(2-methoxyethoxy)-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
2,5-dioxo-6-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-3-yl)benzoic acid
3-(2-hydroxyphenyl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-pyrazole-5-carboxamide
5-methyl-3-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1H-indole
4-(4-butanoylpiperazin-1-yl)-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2,4-dimethylphenyl)-3-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)propanamide
3-[1-(5-ethylpyrimidin-2-yl)piperidin-3-yl]propanamide
(3-{2-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-[(3R,4S)-1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-4-propylpyrrolidin-3-yl]propane-1-sulfonamide
4-[1-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)ethyl]morpholine
N-phenyl-3-{1-[2-(3-phenylpiperidin-1-yl)acetyl]piperidin-4-yl}propanamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-methyl-1-(quinolin-3-yl)-1H-pyrazole-3-carboxylic acid
1-cyclopentyl-4-(2,6,8-trimethylquinoline-4-carbonyl)piperazin-2-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethan-1-one
1-[3-(diethylamino)pyrrolidin-1-yl]-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
methyl 1-({2-[4-(methoxycarbonyl)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)piperidine-2-carboxylate
2-{1-[(5-fluoro-2-methylphenyl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
2-methoxy-N-{2-[3-(morpholin-4-ylmethyl)phenyl]phenyl}acetamide
(3S,4S)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-(naphthalen-2-yl)piperidin-3-ol
5-(4-chlorophenyl)-N-[(2,6-difluoro-3-methylphenyl)methyl]-1,2,4-triazin-3-amine
1-{1'-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-(3-benzamido-4-methoxyphenyl)-3-chloropyridine-4-carboxamide
9-ethyl-1-methyl-4-(quinolin-8-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-methyl-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-methyl-1-{2-[5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}propan-1-one
1-[(2E)-2-methylbut-2-en-1-yl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[(3-methylphenyl)methyl]piperazine
(3aS,6aR)-5-[2-(2-fluorophenyl)acetyl]-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(5-methyl-1H-pyrazol-1-yl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(1R,3S)-3-methoxy-7-[2-(phenylamino)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
2-[cyclopentyl(methyl)amino]-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one