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ethyl 1-ethyl-5-[2-(pyridin-2-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2S)-2-{1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl}pyrrolidine-1-carboxamide
1-[1'-(1H-indole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
1-(5-fluoropyrimidin-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-methyl-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
6-(3-chlorophenyl)-N-(1-hydroxy-3-methylbutan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
1-ethyl-4-{4-[4-(4-methoxypiperidin-1-yl)piperidin-1-yl]benzoyl}piperazine
2-{2-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)quinolin-8-yl]-2-(morpholin-3-yl)acetamide
1-(2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}ethyl)piperidin-2-one
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]quinoline
3-[(4-methoxyphenyl)methyl]-1-methyl-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(4-methoxy-2-methylphenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[2-({[1-(3,4-dimethylphenyl)propyl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
N-(1-methoxypropan-2-yl)-5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-(morpholin-4-yl)butan-1-one
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
methyl 2-[4-(4-cyclopentylpyrimidin-2-yl)-3-methyl-2-oxopiperazin-1-yl]acetate
2-(2-hydroxyethyl)-9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
5-{[(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]methyl}-N-methylfuran-2-carboxamide
7-(4-fluorophenyl)-2-(1,3-thiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)methanesulfonamide
4-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)quinoline
methyl 4-[5-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)furan-2-yl]benzoate
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
2-(4-chloro-2-methylphenoxy)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
ethyl 4-{[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}piperidine-1-carboxylate
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(prop-2-en-1-yloxy)benzamide
dimethyl[2-(2-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
1-ethyl-N-[3-(methylsulfanyl)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
8-[2-(3-hydroxyphenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(5-methylfuran-2-yl)methyl]-3-[1-(morpholine-4-carbonyl)piperidin-3-yl]propanamide
N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-[3-(trifluoromethyl)phenyl]urea
7-[(3-methylphenyl)methyl]-2-(1-propylpiperidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(carbamoylmethyl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-(quinoxaline-6-carbonyl)pyrrolidine-3-carboxylic acid
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2,2-dimethylcyclopropane-1-carboxamide
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-methylpiperazine-1-carboxamide
2-(2,4-difluorophenyl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
5-(5-methyl-1,3-oxazol-4-yl)-3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-[1-(3-methoxyphenyl)ethyl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
(1-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
5-(methoxymethyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
4-{[(3-methoxyphenyl)methyl]amino}-5-methyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-{2-[2-(3-hydroxyphenyl)-1H-imidazol-1-yl]ethyl}-4-methoxybenzene-1-sulfonamide