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N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-(piperidin-3-yl)benzamide
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
5-[2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-2-methoxyphenol
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
1-[2-(dimethylamino)ethyl]-5-(oxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-cyclopropyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}imidazolidin-4-one
5-{[benzyl(methyl)amino]methyl}-N-[(2S)-1-hydroxypropan-2-yl]-1,2-oxazole-3-carboxamide
6-(4-carbamoylpiperidin-1-yl)-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-(3-hydroxypropyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-(6-phenoxypyridin-3-yl)urea
5-methoxy-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-oxo-1,4-dihydropyridine-2-carboxamide
2-methyl-1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-[4-({[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}methyl)phenyl]butanamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-2-amine
4-{[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzonitrile
3-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]-N-methylbenzamide
N-[4-({[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methylbenzamide
(2R,6R)-4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-(1H-indol-3-yl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
(1R,3S,5S)-8-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
3-[2-(1H-imidazol-4-yl)ethyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
5-chloro-2-hydroxy-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]benzamide
[2-fluoro-5-(5-methoxypyridin-3-yl)phenyl]methanol
2,2-dimethyl-N-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-propylpiperidine
methyl 3-{[(2,3-dimethyl-1H-indol-7-yl)formamido]methyl}-5-[2-(thiophen-3-yl)acetamido]benzoate
(2S,4S)-4-amino-N-[(3-methoxyphenyl)methyl]-1-methyl-N-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
2-(ethylamino)-N-{[5-(4-fluorophenyl)furan-2-yl]methyl}pyrimidine-5-carboxamide
1-(2-amino-6-methoxypyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(2-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-methyl-5-{5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
9-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4R)-3-hydroxy-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]pyridine-2-carboxamide
3-[4-(methylsulfanyl)benzoyl]-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
N,N-dimethyl-1-[(6-methylpyridin-2-yl)methyl]azepan-4-amine
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
6-(2-methoxyphenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyridazin-3-amine
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-6-(thiophen-2-ylsulfanyl)pyrimidin-2-amine
4-{[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
2-[(1H-imidazol-4-ylmethyl)(thiophen-3-ylmethyl)amino]butan-1-ol
3,3-dimethyl-1-[(3S,4R)-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-4-methyl-2-(piperidin-1-yl)pyrimidine
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]propan-1-one
N-(3-{[(2-methoxybutyl)carbamoyl]methoxy}phenyl)propanamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-benzyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-[3-(1H-pyrazol-3-yl)phenyl]-2-(trifluoromethyl)pyridine