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2-[(2-methylphenyl)sulfanyl]-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
1-[(4-methoxyphenyl)methyl]-4-(1-methyl-2-oxoimidazolidine-4-carbonyl)piperazin-2-one
(3aR,5S,6S,7aS)-2-[(2-cyclohexylpyrimidin-5-yl)methyl]-octahydro-1H-isoindole-5,6-diol
4-[(2-fluorophenyl)methyl]-1-(1,3-thiazol-2-ylmethyl)piperidine
8-[4-(benzyloxy)butyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-{5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]furan-2-yl}-1H-pyrazole
4-[(1-acetylpiperidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
methyl 4-{[3-(diethylcarbamoyl)piperidine-1-carbonyl]amino}-3-methylbenzoate
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-N-propyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[(3aS,6aS)-2-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
7-(2-methoxyethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-methyl-1-(3-methylphenyl)-4-[2-(pyrrolidin-1-yl)benzoyl]piperazin-2-one
(2Z)-3-(3-fluorophenyl)-1-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}prop-2-en-1-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}propan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]butan-1-one
3-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridazine
(1S,5R)-3-benzyl-6-(2-methyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)piperidin-3-amine
N-[(3-methoxyphenyl)methyl]-1-[3-(1,3-oxazol-5-yl)phenyl]piperidin-4-amine
1-(3,5-dimethylphenyl)-4-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperazin-2-one
1-(1-cycloheptylpiperidin-3-yl)-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2-methylphenoxy)ethan-1-one
N-cyclopropyl-5-methyl-4-{[(5-methylfuran-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-{2-hydroxy-3-[2-methoxy-4-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
6-butyl-2-[4-(piperidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
4-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4-methylpiperidine
4-{2-[(4-methylpyrimidin-2-yl)oxy]hex-5-en-1-yl}-1,4-oxazepane
2-{2-[1-(2-chloro-4-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-ethyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-propyl-1H-pyrazole-3-carboxamide
[(1-cyclohexylpiperidin-3-yl)methyl][(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](pyridin-3-ylmethyl)amine
1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
3-(1-butyl-1H-imidazol-2-yl)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
2-({6-[3-(4-phenylbenzoyl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
(3S)-1-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N,N-dimethylazepan-3-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1,2-oxazole-3-carboxamide
6-chloro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethylimidazo[1,2-a]pyridine-3-carboxamide
8-(1H-indol-3-ylmethyl)-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4S)-1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-4-phenylpyrrolidin-3-amine
3-(1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
8-[(3-carboxy-1H-pyrazol-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,8aR)-6-(1,3-benzothiazole-5-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
(3R,9aR)-8-(4-methylbenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,6-dimethyl-2-oxo-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-tert-butyl-4-(1-ethyl-1H-1,2,4-triazol-5-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4aR,7aS)-4-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-(azepane-1-carbonyl)-N-[(2,3-dimethoxyphenyl)methyl]-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
N,N-diethyl-4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]aniline
5-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one