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1-(2-{1-[3-(pyridin-2-yl)propanoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
3-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
8-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)piperazin-1-yl]-N-ethylacetamide
1-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-5-methyl-1H-1,2,3,4-tetrazole
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,3-dihydroxypropan-2-yl)propanamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-1,3-benzothiazole-5-carboxamide
2-methyl-3-{[4-(oxan-4-yl)piperazin-1-yl]methyl}quinoxaline
1-methyl-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine-2-carboxylic acid
(3R)-1-[6-(methoxymethyl)pyrimidin-4-yl]-3,4,4-trimethylpyrrolidin-3-ol
ethyl 4-({[3-(2-oxopyrrolidin-1-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
4-[4-(3,4-difluorobenzoyl)piperidine-1-carbonyl]-1-ethylpyrrolidin-2-one
4-[(cyclopropylmethyl)amino]-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
4-(hydroxymethyl)-1-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]azepan-4-ol
(1S,6R)-9-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
4-{2-[1-(pyrrolidine-1-sulfonyl)piperidin-2-yl]ethyl}phenol
4-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]phenol
(3S,7S)-5-(3-methanesulfonamidopropanoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-ethyl-1H-pyrazole-5-carboxamide
1-[(2-{[(6-methoxypyrimidin-4-yl)amino]methyl}phenyl)methyl]pyrrolidin-2-one
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
2-{3-cyclopentyl-5-[(2-oxopiperidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}benzoic acid
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
5-[1-(1-benzofuran-5-carbonyl)pyrrolidin-2-yl]-N-propylthiophene-2-carboxamide
N-[2-({[1-(carbamoylmethyl)-2-methyl-1H-indol-3-yl]methyl}amino)ethyl]acetamide
N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-propylpiperidin-4-amine
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-(2-{1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(piperidin-1-yl)acetamide
8-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-N-[(1-ethylpyrrolidin-3-yl)methyl]-3-methyl-1H-pyrazole-4-sulfonamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(methylsulfanyl)propanamide
1-{[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-cyclobutaneamido-N-cyclohexyl-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
3-[6-(cyclopentylamino)pyridazin-3-yl]phenol
1-cyclopropyl-N-[2-(2-methoxynaphthalen-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
5-oxo-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-7-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(cyclopropylmethyl)-8-[2-(2-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-cyclohexyl-3-[(4-hydroxy-2-phenylpyrimidin-5-yl)formamido]propanamide
1,3-dimethyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2-methylpropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide