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5-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}-2-(2-methylphenyl)pyrimidine
1-(4-phenyl-1,4-diazepan-1-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-methyl-1H-indol-3-yl)acetamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(2-methylpropanoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
[3-(2-methoxyethyl)-1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]methanol
(2S,4R)-4-amino-N,N-diethyl-1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)pyrrolidine-2-carboxamide
1-{2-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
8-(2-ethylpyridine-4-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
5-(2-{3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}phenoxy)pyrimidine
1-[3-({[2-(dimethylamino)ethyl]({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)amino}methyl)phenyl]ethan-1-one
3-phenyl-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperazine
4-(5-fluoro-2-methylphenyl)-6-methylpyrimidin-2-amine
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(5-methylpyridine-3-carbonyl)-1,4-diazepane
1-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
(1S,5R)-6-benzyl-3-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethan-1-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
(1S,5R)-3-benzoyl-N-(3,5-dimethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[2-(dimethylamino)ethyl]-5-[(2S)-pyrrolidine-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4,4-difluoro-1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidine
(3S,4S)-4-(4-fluorophenyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-ol
3-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-1-(2-methoxyethyl)-6-methyl-1,2-dihydroquinolin-2-one
8-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
1-[9-acetyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(pyrazin-2-yl)ethan-1-one
6-{[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}-2-methylpyrimidin-4-ol
2-({6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidin-4-yl}amino)ethan-1-ol
8-(2-cyclopropylacetyl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3-cyclohexylpyrrolidine-1-carbonyl)-2-(4-methoxyphenoxymethyl)-1,3-oxazole
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-[(4aR,8aS)-1-benzoyl-decahydro-1,6-naphthyridin-6-yl]-2-phenoxyethan-1-one
1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
3-(5-fluoro-2-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
(3R)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(3aR,7aS)-2-{2-[(6-ethylpyrimidin-4-yl)oxy]hex-5-en-1-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-2,6-dimethylpyridine-4-carboxamide
(4aR,7aS)-1-ethyl-4-{pyrazolo[1,5-a]pyridine-7-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-fluoro-4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-benzyl-5-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}pyrimidin-2-amine
1-{3-[3-(pyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
1-[2-(2-hydroxyethyl)piperidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-[2-(1H-pyrazol-1-yl)ethyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide
1-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholin-3-yl}acetyl)piperidine-4-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trimethylbenzamide
1-methyl-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
4-[3-(pyrrolidin-1-ylmethyl)phenyl]aniline
(1R,5S,8S)-8-methoxy-N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-3-azabicyclo[3.2.1]octane-3-carboxamide