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1-{2-[4-(4-fluorophenoxy)piperidin-1-yl]ethyl}-1H-indazole
N-cyclopropyl-5-(4-methoxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]furan-2-carboxamide
1-(cyclopent-3-en-1-yl)-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
4-hydroxy-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N,N-dimethyl-5-[methyl(naphthalen-1-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenol
2-{5-[3-(1,1-dioxo-1λ6-thiomorpholin-4-yl)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)piperazine
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
2-(methylamino)-N-[3-(4-methylbenzenesulfonamido)propyl]pyridine-4-carboxamide
[(3R,4R)-1-(7-fluoro-2-methylquinoline-4-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(1-ethyl-5-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
1-{1-[2-(thiophen-2-yl)azetidine-1-carbonyl]cyclopentyl}pyrrolidine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}pyrimidine
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
{1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
1-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-(thiophen-3-ylmethyl)piperazine
5-methyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]pyrazine-2-carboxamide
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
2-ethyl-4-[6-(6-methoxypyridin-3-yl)pyridine-3-carbonyl]-1-(propan-2-yl)piperazine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(1-propylpiperidin-4-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-methoxy-1-[6-methyl-5-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]propan-1-one
1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-{2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N4-(furan-2-ylmethyl)-6-(propan-2-yloxy)pyrimidine-2,4-diamine
4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyridine
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
3-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
1-{[4-(furan-2-yl)phenyl]methyl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-imidazol-1-yl)-N-methylbenzamide
1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
3-(ethylsulfanyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
6-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
4-(2-{1-[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]piperidin-2-yl}ethyl)morpholine
(1R,2R,4R)-N-[2-(1,3-benzoxazol-2-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[3-(3-oxopiperazin-1-yl)propyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
methyl 2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
2-{4-[(3,5-difluorophenyl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
methyl 3-(4-{1-benzyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrazol-1-yl)propanoate
1-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
5-(4-methyl-1,4-diazepan-1-yl)-2-[3-(pyridin-3-yl)propyl]-2,3-dihydropyridazin-3-one
N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[2-(methylsulfanyl)ethyl]amine
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidine