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1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(oxan-4-yl)piperazine
ethyl 2-[methyl(5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyrimidin-2-yl)amino]acetate
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)amine
2-(3-benzyl-1H-1,2,4-triazol-5-yl)-3-methylpyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]thiophene-2-carboxamide
2-(1H-1,2,4-triazol-1-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-hydroxypropan-1-one
5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidin-2-yl}-N-(furan-2-ylmethyl)thiophene-2-carboxamide
4-[(dimethylamino)methyl]-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]azepan-4-ol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-5-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-[(4aR,8aR)-7-(2,1,3-benzoxadiazol-4-ylmethyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(1R,5S,8R)-3-[(2-methoxynaphthalen-1-yl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
3,6-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
methyl (1R,3R,3aR,6aS)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-3-[2-(1H-pyrazol-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
{1-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]piperidin-4-yl}(pyridin-2-yl)methanol
(3aR,6aS)-5-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-cyclohexylethan-1-one
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
2-methoxy-N-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}benzamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-(2-methoxyphenoxy)azetidine
1-(2-methylphenyl)-4-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperazin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
(1S,5R)-3-(3-phenylpropyl)-6-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]phenol
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[(dimethylamino)methyl]-1,3-thiazole-4-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N4-methyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine-2,4-diamine
2-{[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(propan-2-yl)piperidine
1-[1-(2,3-dihydro-1H-isoindole-1-carbonyl)piperidin-4-yl]piperidin-4-ol
(4aS,8aR)-6-(2-ethoxyacetyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
3-({[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)piperidin-3-ol
(2S,4R)-N,N-diethyl-1-methyl-4-{5-[(methylsulfanyl)methyl]furan-2-amido}pyrrolidine-2-carboxamide
3-(propan-2-yl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-5-carboxamide
methyl 2-(benzylsulfamoyl)-6-(thian-4-yl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-({[(3R,4R)-4-(hydroxymethyl)-1-{2-[(4-methylphenyl)methyl]benzoyl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(2,3-dihydro-1H-inden-5-yl)-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]urea
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2,6-dimethoxybenzamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(4-methoxybenzoyl)piperazine
7-methyl-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[(5-chloro-2-fluorophenyl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
6,7-dimethoxy-2-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-methyl-1,2,3,4-tetrahydroisoquinoline
3-[(3R,4S)-1-[1-(2-methylphenyl)piperidin-4-yl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-(2H-1,3-benzodioxol-5-yl)-5-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine-1-carboxamide
N-cyclohexyl-3-({[4-(1,3-thiazol-4-yl)phenyl]carbamoyl}amino)propanamide
1-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(furan-2-yl)propan-1-one
(2R)-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxy-2-phenylethan-1-one