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[(3S,5R)-5-[(dimethylamino)methyl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]methanol
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-methylphenyl)-1,4-diazepane
2,3-dimethoxy-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-3-(thiophen-2-yl)urea
5-{5-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
N-[4-(furan-2-yl)butan-2-yl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
1-[4-(2-benzylmorpholin-4-yl)-4-oxobutyl]piperidin-2-one
3-methyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazine
1-methyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N'-(2,3-dimethylphenyl)-N-(1H-indol-4-ylmethyl)propanediamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetic acid
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-fluoro-5-sulfamoylbenzamide
2-chloro-N,N-dimethyl-5-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}carbamoyl)amino]benzamide
3-(azepane-1-sulfonyl)-5-(2,6-dimethoxyphenyl)benzoic acid
8-fluoro-2-({[1-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)quinolin-4-ol
3-(2-methylphenyl)-5-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazole
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
2-{[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}acetic acid
2-amino-6-butanoyl-4-[6-(dimethylamino)pyridin-3-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
9-(4-methanesulfonylphenyl)-6-methyl-9H-purine
2-methyl-5-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrazine
3-{5-[2,5-dimethyl-1-(propan-2-yl)-1H-pyrrol-3-yl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1-methylpiperazine-2-carboxylic acid
2-{1-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-N-methylformamido}-N,2-dimethylpropanamide
N,2,5-trimethyl-N-(pyrazin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(4-fluorophenyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-amine
(3R,4R)-4-ethyl-1-[2-(2-phenylethoxy)benzoyl]piperidine-3,4-diol
(3S,4R)-1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
4-[(2-methyl-1H-imidazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
[(4-methanesulfonylphenyl)methyl](methyl)[1-(pyridin-2-yl)propan-2-yl]amine
4-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[2-(4-hydroxyphenyl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
5-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]-2,4-dimethylpyridine
4-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}morpholine
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-(2-methylpyrimidin-4-yl)piperidine-1-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
3-(3-fluorophenyl)-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-cyclopropyl-3-(furan-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
7-chloro-3-{[(2,2-diphenylethyl)amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}diphenylmethanol
5-[4-(3-chlorophenyl)-3-oxopiperazine-1-carbonyl]-2-cyclopropyl-3,4-dihydropyrimidin-4-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(4-ethylphenoxy)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
N-methyl-2-(2-methyl-1H-imidazol-1-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
2-(azocan-1-yl)-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
[(4-ethyl-1,3-thiazol-2-yl)methyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
1-(2-methylphenyl)-3-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
methyl (2S,3S)-2-({1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-yl}amino)-3-methylpentanoate
[3-(2-methoxyethyl)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]methanol