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5-methyl-N4-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrimidine-2,4-diamine
2,8-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]quinoline-4-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N3-[(3-phenylphenyl)methyl]piperidine-1,3-dicarboxamide
2,5-dimethyl-3-(4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-1-yl)pyrazine
[(4aS,8aR)-6-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
6,7-dimethoxy-2-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(oxan-4-ylmethyl)amine
8-(5-methyl-1H-indazole-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(5-{[(butan-2-yl)(3-phenylprop-2-yn-1-yl)amino]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-[(3-methoxyphenyl)sulfanyl]acetamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-ethyl-1'-{thieno[3,2-d]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
4-{[2-(methanesulfonamidomethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}benzoic acid
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
5-methoxy-9-(5-propyl-1,3,4-oxadiazol-2-yl)-1-oxa-9-azaspiro[5.5]undecane
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-(3-{1-[(5-fluoro-2-methylphenyl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
5-(azepane-1-carbonyl)-N-[1-(2-chlorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[(piperidin-3-yl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}pyrrolidine-1-carboxamide
2-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane
1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-[(dimethylamino)methyl]piperidin-4-ol
2-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
N3-tert-butyl-1-cyclohexyl-N5-[(1-methylpiperidin-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 2-{3-[3-(3-cyanophenyl)phenyl]-1H-pyrazol-1-yl}acetate
N-[3-(cyclohexyloxy)propyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3-chloro-2-methylphenyl)methyl]-2-[methyl(piperidin-4-yl)amino]acetamide
8-(5-methoxyfuran-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-cyclopentyl-4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-{4-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-(2,6,8-trimethylquinoline-4-carbonyl)azetidine-2-carboxylic acid
N-{[2-(diethylamino)pyridin-3-yl]methyl}-3-ethyl-1,2-oxazole-5-carboxamide
5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-methyl-1-(4-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
8-[(3-hydroxyphenyl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(3-methoxyphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2,4-triazin-3-amine
2-(4-fluorophenyl)-2-hydroxy-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
[2-(3-chloro-5-methylpyridin-2-yl)phenyl]methanol
2-(dimethyl-1,3-thiazol-5-yl)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]acetamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-N'-(4-methylphenyl)propanediamide
7-(1-benzothiophene-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[2-(3-methoxyphenoxy)ethyl]-4-(4-methylpiperidine-4-carbonyl)piperazine
1-[3-(2-methoxyethoxy)phenyl]-3-methyl-3-(pyrazin-2-ylmethyl)urea
(2,3-dihydro-1-benzofuran-5-ylmethyl)[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
(4aS,8aR)-6-(2-amino-4-methylpyrimidine-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one