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1-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)-2-phenoxyethan-1-one
2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1,2,3,4-tetrahydroisoquinolin-4-ol
N-{3-[({[5-(3-chlorophenyl)furan-2-yl]methyl}amino)methyl]-5-(dimethylcarbamoyl)phenyl}pyridine-2-carboxamide
(4aS,8aR)-2-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-decahydroisoquinoline
N-cyclopropyl-1-{2-[1-(2-methylbenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3-carboxamide
1-{[5-(1-benzothiophen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
3-(2-fluorophenyl)-5-(oxan-4-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[2-(furan-2-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(4aS,8aS)-2-[(2,4-diethoxy-3-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-pyrrol-1-yl)propan-1-one
N-ethyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
4-{[2-(cyclohexylcarbamoyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
(4aR,7aS)-1-ethyl-4-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,6R)-9-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
(2S,4S)-4-amino-1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-N-methylpyrrolidine-2-carboxamide
N-[(2S)-1-hydroxybutan-2-yl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
2-(4-chloro-1H-pyrazol-1-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propan-1-one
N-(2-chlorophenyl)-3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propanamide
4-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-[(3-acetylphenyl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
3-{1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}phenol
1-(4-fluorobenzenesulfonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
6,7-dimethoxy-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinazolin-4-amine
1-(cyclohex-3-ene-1-carbonyl)-4-(4-fluorophenoxy)piperidine-4-carboxylic acid
1-[4-(4H-1,2,4-triazol-4-yl)phenyl]azepane
2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4-methylphenol
7-[(2,3-difluorophenyl)methyl]-2-(pyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(2S)-N1-[2-(2-ethoxyethoxy)phenyl]pyrrolidine-1,2-dicarboxamide
1-methyl-9-{[4-(2-methylphenyl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
9-[(2-butyl-1H-imidazol-4-yl)methyl]-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
N-(furan-2-ylmethyl)-N-methyl-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[(4-chlorophenyl)methyl]-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
(3S,4R)-4-methyl-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine-3,4-diol
2-[4-(4-fluorophenyl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
2-chloro-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-6-fluorobenzamide
1-tert-butyl-3-[2-(methylsulfanyl)ethyl]-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
(2S,4R)-4-amino-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)pyrrolidine-2-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-(4-fluorophenyl)-1H-pyrazol-1-yl]acetamide
3-({1-ethyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-3,4-dihydroquinazolin-4-one
7-(3-chlorophenyl)-4-(5-propyl-1,2,4-oxadiazol-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(1,2,5-thiadiazole-3-carbonyl)piperazine
2-(5-acetylthiophen-3-yl)-1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
9-(5-methyl-1,2-oxazole-3-carbonyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-8-(propan-2-yl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(dimethylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-3-phenylpyrrolidin-3-ol
4-(furan-2-ylmethyl)-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-ethyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-methylpyrimidin-4-amine
(3R,4S)-1-cycloheptanecarbonyl-4-cyclopropylpyrrolidin-3-amine