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1-{3-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)benzamide
N1-methyl-N2-[2-(5-methylfuran-2-yl)ethyl]cyclohexane-1,2-dicarboxamide
1-methyl-4-({5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
4-(4-methanesulfonylphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(1R,3s,6r,8S)-4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-azatricyclo[4.3.1.13,8]undecane
6,8-dimethyl-2-({4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
5-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
(3aR,6aR)-2-benzyl-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1,3-dimethyl 5-{[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]amino}benzene-1,3-dicarboxylate
(1R,4S)-2-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carbonyl}-2-azabicyclo[2.2.1]heptane
(1-{[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
1-methyl-3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl]methanol
ethyl 4-[6-oxo-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-1H-pyrazole-3-carboxylate
4-(4-chlorophenoxy)-1-(1H-imidazol-4-ylmethyl)piperidine
4-[(6-chloro-4-{[3-(propan-2-yloxy)propyl]amino}quinazolin-2-yl)methyl]piperazin-2-one
8-{[3-methyl-4-(pyrrolidin-1-yl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(4-fluorophenyl)formamido]-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]propanamide
3-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl)amino}-N-(2-fluorophenyl)propanamide
7-ethyl-2-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-[(2-chlorophenyl)methyl]-4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1H-1,2,3-triazole
4-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}-N-methylbutanamide
2-phenyl-N-[3-(piperidin-1-ylmethyl)phenyl]azetidine-1-carboxamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(4-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
2-[1-(2-methylpropyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl]ethan-1-ol
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
N-[(2-ethoxypyridin-3-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-(2,3-dihydro-1-benzofuran-7-yl)-6,7-dimethoxyquinazolin-4-amine
2-amino-4-(furan-3-yl)-6-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)methyl]piperidin-2-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methylthiophene-2-carboxamide
7-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{1-[5-(hydroxymethyl)furan-2-carbonyl]piperidin-4-yl}pyrrolidin-2-one
5-fluoro-N2,N4,N4-trimethyl-N2-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
2-(2-{[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
8-fluoro-2-(3-propoxypiperidine-1-carbonyl)quinoline
N,N-diethyl-2-[2-(ethylamino)pyrimidin-5-yl]-3,6-dimethylquinoline-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(2,1,3-benzothiadiazol-5-ylmethyl)amine
4-ethenyl-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
ethyl 1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}piperidine-3-carboxylate
4-fluorophenyl (3R,9R)-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxylate
ethyl 1-(but-2-ynoyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-({1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
4-{1-[(3-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-methyl-1-propyl-1H-pyrazole
2-amino-4-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-ethyl-N-methyl-1,2-oxazole-5-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[(2-chloro-6-fluorophenyl)methyl]-5-{[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1H-1,2,4-triazole