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1-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
4-(3-methoxypyridin-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(3R,4S)-4-{[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](ethyl)amino}oxolan-3-ol
3-[1-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-3-yl]benzoic acid
4-methoxy-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
N-[1-(3-methylphenyl)piperidin-4-yl]-1-(pyridin-3-ylmethyl)azepan-3-amine
4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
(4aR,8aS)-6-cyclohexyl-1-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2-[1-(pyrazin-2-yl)piperidin-3-yl]-1H-1,3-benzodiazole
N-(1,3-thiazol-2-ylmethyl)-N-(thiophen-3-ylmethyl)cyclopropanamine
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyridine-3-carboxamide
2-(5-chloro-3-fluoropyridin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-phenyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
(2R)-2-amino-1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-hydroxypropan-1-one
methyl (2S,4R)-1-methyl-4-[(2S)-oxolane-2-amido]pyrrolidine-2-carboxylate
N-(2,3-dihydroxypropyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
2-{9-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(1,8-naphthyridine-2-carbonyl)piperidin-3-ol
2-chloro-N-[2-(2-oxoimidazolidine-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-methoxy-4-[({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
1-[2-methoxy-5-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
2-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
2,3,5-trimethyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-[(4-ethoxyphenyl)methyl]piperazin-2-one
1-({[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]carbamoyl}amino)-N-methylcyclohexane-1-carboxamide
3-(4-methoxyphenyl)-N-{1-[(4-methylphenyl)methyl]cyclopropyl}-1H-pyrazole-5-carboxamide
N-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-[2-(ethylsulfanyl)ethyl]cyclohexanamine
2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-4-(3,3,3-trifluoropropyl)pyrimidine
3-(3,3-diphenylpiperidine-1-carbonyl)-1λ6-thiolane-1,1-dione
N-[(3,4-difluorophenyl)methyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
2,6-dioxo-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-methyl-5-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(2-methoxyphenyl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
4-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2-(trifluoromethyl)morpholine
N-[1-(1H-indol-5-yl)ethyl]-6-(methoxymethyl)pyridine-2-carboxamide
8-(1H-indol-5-ylmethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-chloro-2-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-1H-indole
2-{3,5-dimethyl-4-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]-1H-pyrazol-1-yl}acetic acid
5-(3-fluorophenoxymethyl)-N-[1-(hydroxymethyl)cycloheptyl]-1H-pyrazole-3-carboxamide
2-({[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)quinolin-4-ol
N-butyl-N-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
2-[1-(1-benzothiophene-5-carbonyl)piperidin-2-yl]pyridine
[3-(4-fluorophenoxy)propyl](methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
N-[(3R,4S)-4-cyclopropyl-1-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl]-1-(methoxymethyl)cyclopropane-1-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-cyclopentyl-4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
3-ethyl-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-indole-2-carboxamide