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1-[(5-ethylpyridin-2-yl)methyl]-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine
1-[(1-methylpiperidin-3-yl)methyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
5-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4-methyl-1,3-oxazole
1-(cyclopropanesulfonyl)-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[3-(1H-imidazol-2-yl)benzoyl]-1-(3-methoxyphenyl)piperazin-2-one
2-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
1-{6-hydroxy-4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1,4-diazepan-1-yl}-3-methoxypropan-1-one
2-methyl-N-{3-[(pyridin-3-yl)amino]propyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(1S,2R)-2-carbamoylcyclopentyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(2-{[4-(1-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
methyl 1-(benzyloxy)-2-oxo-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
3-{4-[4-(pyrrolidin-1-yl)piperidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}-1H-indole
2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxylic acid
4-(5-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
3-butyl-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-methylpiperazin-2-one
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-N-(2,4-dimethoxyphenyl)propanamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
2-methyl-N-[(5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl)methyl]-1,3-thiazole-4-carboxamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{1-[1-(thiophene-2-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
3-{[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-(4-chloro-1H-pyrazole-3-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
N-[(4-methoxyphenyl)methyl]-1,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-(piperidin-3-ylmethyl)-N-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(cyclopropylmethyl)-1-[3-(2-methoxyphenyl)propanoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(2S,4S)-N-ethyl-4-(5-methylthiophene-2-amido)-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
5-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]quinoxaline
(3R,4R)-1-(4-methoxypyrimidin-2-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(2R,3R)-3-{[3-(2-fluorophenyl)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(4-fluorophenyl)-1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-amine
1-benzyl-4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-2-one
2-[({1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
N-{[1-(methoxymethyl)cyclopentyl]methyl}-4-(piperidin-3-ylmethyl)benzamide
1-(4-ethylpiperazin-1-yl)-3-[3-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
(1R,6S)-9-methyl-3-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3,9-diazabicyclo[4.2.1]nonane
(2R,4R)-4-hydroxy-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]pyrrolidine-2-carboxamide
6-ethyl-N,2-dimethyl-N-[1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
4-(3-fluorophenoxy)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
(3S,4R)-4-(3-methoxyphenyl)-1-(oxane-4-carbonyl)pyrrolidine-3-carboxylic acid
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(4-fluorophenoxymethyl)piperidine
2-(methylsulfanyl)-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}azepane
(2S)-3-methyl-2-{[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}butanamide
5-benzyl-1-(4-methylphenyl)-4-[(3E)-pent-3-enoyl]piperazin-2-one
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
1-[(4aR,8aS)-6-cyclopropanecarbonyl-decahydro-1,6-naphthyridin-1-yl]-2-phenoxypropan-1-one