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2-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
N-[(3R,4S)-4-cyclopropyl-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-3-yl]ethane-1-sulfonamide
4-({[4-(pyridin-2-yl)pyrimidin-2-yl]amino}methyl)benzene-1-sulfonamide
1-(2-methoxyethyl)-4-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperazine
2-(1-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}piperidin-2-yl)acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-(1-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
(1R,5S,6S)-6-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(2,4-dimethoxyphenyl)-3-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]propanamide
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(propan-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(3,6-dimethylpyrazin-2-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(quinolin-8-ylmethyl)-2,7-diazaspiro[4.5]decane
N-[2-(methylsulfanyl)ethyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-(1-hydroxybutan-2-yl)-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamide
1-benzyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-[3-(4-fluorophenoxy)piperidin-1-yl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
8-(2-amino-6-methylpyrimidin-4-yl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)quinoline
1-{[1-ethyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}pyridine
N-[2-(1-methylpiperidin-3-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(adamantan-1-yl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]acetamide
3-[(3-methoxyphenyl)methyl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-methyl-4-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}morpholine-2-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
5-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2-methoxypyrimidine
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
1-cyclobutanecarbonyl-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-benzyl-3-ethyl-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1,4-diazepan-5-one
4-[(2S)-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carbonyl]morpholine
2-cyclopropanecarbonyl-8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-ethyl-4-methyl-N-(5-methyl-2-pentanamidophenyl)-1,3-oxazole-5-carboxamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
1-(3-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(5-propylfuran-2-yl)methyl]piperidine
2-{[2-amino-6-(2,4,6-trimethylphenyl)pyrimidin-4-yl]amino}ethan-1-ol
3-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5-methoxy-3,4-dihydroquinazolin-4-one
4-phenoxy-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
methyl[2-(2-methyl-1H-imidazol-1-yl)propyl][(4-methyl-1H-imidazol-2-yl)methyl]amine
6-fluoro-N-methyl-N-(2-methylpropyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide