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1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
1-(2-phenylethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(1,2,3,6-tetrahydropyridin-4-yl)ethan-1-one
1-[(2,6-difluorophenyl)methyl]-2-(1H-imidazol-4-yl)-1H-imidazole
4-{[4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
2-{4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-imidazol-5-yl}quinoline
{4-[(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
5-(methoxymethyl)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)furan-2-carboxamide
(2R,6R)-10-methoxy-4-[2-oxo-2-(piperidin-1-yl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-methoxy-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
3,5-difluoro-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pyridine-2-carboxamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
5-(2,5-dihydro-1H-pyrrol-2-yl)-1-(4-methoxyphenyl)-3-phenyl-1H-1,2,4-triazole
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(4-methylpiperazin-1-yl)benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-fluoro-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[(3-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-yl)benzoic acid
6-(4-fluorophenyl)-2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
5-ethyl-2,3-dimethyl-N-[2-(oxan-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-3-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[4-(2-methyl-1H-imidazol-1-yl)butan-2-yl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(3,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[(3S,4R)-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
3-(3-methoxyphenyl)-N-[2-(methylsulfamoyl)ethyl]-1H-pyrazole-5-carboxamide
2-[3-(3-chlorophenyl)-4-methyl-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
1-[1-(1-{[4-(pyridin-2-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
N-[4-methyl-2-(1-methyl-1H-pyrazol-4-yl)phenyl]propanamide
3-{[({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
3-methyl-N-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}pyridin-2-amine
5-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-N,N-dimethylpyrimidin-2-amine
(1R,5R)-6-(cyclopropylmethyl)-3-(4-methoxypyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
5-[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-methoxy-2-methylpropan-1-one
2-(3-chloro-4-hydroxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
5-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
9-methoxy-7-[4-(methylsulfanyl)phenyl]-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
dimethyl(2-{2-[1-(quinoline-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-(1,3-benzothiazol-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[4-(aminomethyl)phenyl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-[4-(thiophen-3-ylmethyl)morpholin-3-yl]acetic acid
1-ethyl-N-[2-(furan-2-yl)ethyl]piperidine-2-carboxamide
N-[(4-chlorophenyl)(pyridin-3-yl)methyl]-5-fluoroquinazolin-4-amine
[1-(2-aminopyridine-4-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3,3,3-trifluoropropan-1-one
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide