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(4aR,7aS)-1-(cyclopropylmethyl)-4-(quinolin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}imidazo[1,2-a]pyridine-6-carboxamide
(1S,4S)-2-[4-(morpholin-4-yl)benzoyl]-2,5-diazabicyclo[2.2.1]heptane
(1S,2R)-N1-(3-methoxypropyl)-N1-(1-methylpiperidin-4-yl)-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
6-ethyl-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-2-methylquinoline-4-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{2-[(4-methyl-1,2,3-thiadiazol-5-yl)sulfanyl]ethyl}acetamide
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-methyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
2-amino-6-(3,5-dimethylphenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
5,6-dimethyl-2-[3-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
4-{[1-(5-ethylpyrimidin-2-yl)piperidin-3-yl]methyl}morpholine
5-methyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-(2-hydroxy-3-methoxypropyl)-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(ethylsulfanyl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-{[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]methyl}acetamide
N-(2-methoxyethyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
(3aS,6aS)-2-cyclopentyl-5-[2-(2,4-difluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-hydroxy-1-(2-phenylquinazolin-4-yl)piperidine-4-carboxylic acid
3-({[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-6,8-dimethyl-1,2-dihydroquinolin-2-one
N-[(2R,4S,6S)-2-ethyl-6-(2-phenylethyl)oxan-4-yl]benzamide
1-(3-ethyl-1,2-oxazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N,1-diethyl-N-(oxan-4-ylmethyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1'-[5-(methoxymethyl)furan-2-carbonyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
5-fluoro-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
1-cyclopentanecarbonyl-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,4,7-trimethyl-1H-indole
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4-methylpyrimidine-5-carboxamide
8-(3-ethyl-1H-pyrazole-4-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]-N-(1,2,3-thiadiazol-5-yl)benzamide
(3aR,6aR)-2-[3-(2-methoxyphenyl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}pyridine-3-carboxylate
3-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}phenol
3-(1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidin-3-yl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-{[(2-chlorophenyl)methyl]carbamoyl}ethyl)-3-ethylpiperidine-3-carboxylic acid
3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-[3-(methylsulfanyl)phenyl]urea
N,8-dimethyl-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
(4aS,8aR)-6-(2,4-dimethylpyrimidine-5-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-4-methoxy-2-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]benzamide
6-(4-chlorophenyl)-N-[2-(oxan-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(2-methoxyethyl)-1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-(dimethylamino)-8-(2-oxo-1-phenylpyrrolidine-3-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
4-(1H-pyrazol-4-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
3-(1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)-N-(3-methoxyphenyl)propanamide
6-methoxy-N-[(6-methoxy-2H-chromen-3-yl)methyl]pyridin-3-amine
8-[(1R,3S)-3-aminocyclohexanecarbonyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one