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N-(2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}quinolin-6-yl)acetamide
N-[1-(1H-imidazol-2-yl)ethyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]acetamide
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(piperidin-3-ylmethyl)amine
2-(4-chloro-2-methylphenoxy)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[2-(pyridin-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(cyclohexylmethyl)-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazole
1-[(2R,3R)-3-[ethyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-benzyl-4-propyl-1,4-diazepan-5-one
2-acetyl-8-phenylmethanesulfonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-cycloheptyl-4-[2-(methylsulfanyl)phenoxy]piperidine-4-carboxylic acid
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
N-ethyl-5-[4-(thiophen-3-ylmethyl)piperazine-1-carbonyl]pyrimidin-2-amine
N-[(3-fluoro-4-methylphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
4-{4-[6-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}benzonitrile
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
1-[3-(azetidine-1-carbonyl)benzenesulfonyl]-2-methyl-1,4-diazepan-5-one
1-(cyclohexylmethyl)-N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(pyridin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-benzyl-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
N-(2-methoxyethyl)-N-(naphthalen-1-ylmethyl)-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
(2S,4S)-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
3-{2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-4-ethyl-4H-1,2,4-triazole
3-[1-methyl-5-(1-methyl-5-phenyl-1H-pyrazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
7-[(3-methylphenyl)methyl]-2-[2-(1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylfuran-2-carboxamide
(2R,3S,6R)-5-[(5-ethylpyridin-2-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,6S)-N-(4-cyano-2,5-difluorophenyl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N-methyl-5-{[methyl(2-phenylethyl)amino]methyl}-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-(furan-2-yl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]propan-1-one
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(3-phenylpiperidin-1-yl)acetamide
4-{2-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]ethyl}phenol
3-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N,N-dimethylpyrazin-2-amine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-4-methoxyphenol
2-amino-7-[2-(1H-indol-3-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(naphthalen-1-yl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-[4-(2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethoxy)phenyl]propan-1-one
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine
benzyl[(4-methyl-1,3-thiazol-5-yl)methyl]{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine
ethyl 4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazine-1-carboxylate
(2E)-N-[2-(2-chloro-6-methoxyphenyl)phenyl]but-2-enamide