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2-(3-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}-1H-indol-1-yl)acetamide
3-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)carbamoyl)methyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
2-methyl-5-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}pyrazine
[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl][1-(4-methylpiperazin-1-yl)propan-2-yl]amine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(1H-indol-1-yl)propyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
6-(methoxymethyl)-N,1-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{3-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2,5-dimethylpyrazine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-ethoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
N-{2-[2-(trifluoromethyl)phenyl]ethyl}-6-azaspiro[2.5]octane-1-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,5,6-trimethylthieno[2,3-d]pyrimidin-4-amine
3-{1-[(3,3-diphenylpropyl)carbamoyl]-6-azaspiro[2.5]octane-6-carbonyl}pyridin-1-ium-1-olate
4-chloro-1-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
4-ethoxy-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidin-2-amine
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-6-(methoxymethyl)pyridine-2-carboxamide
1-(2-aminoethyl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-benzyl-3-ethyl-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1,4-diazepan-5-one
2,2,3,3-tetramethyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}cyclopropane-1-carboxamide
N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}-1,3-thiazole-5-carboxamide
2-{methyl[(4-methylphenyl)methyl]amino}-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2,4,6-trimethylphenyl)quinoxaline
3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}propanoic acid
4-methyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-imidazole-2-carboxamide
1-[(4-chloro-3-fluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
N-cyclohexyl-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-propyl-1H-pyrazole-5-carboxamide
5-methyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine
(1S,6R)-9-[3-(2-methyl-1,3-thiazol-4-yl)benzenesulfonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(1R,5S,8S)-3-[(2-chloro-6-fluorophenyl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
N-[(3-methoxyphenyl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-methyl-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroquinoxalin-2-one
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-N-methylpyrrolidine-3-carboxamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
3-({1-[4-(2-oxopiperidin-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
5-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-oxo-4H-pyran-2-carboxamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{2-[2-(trifluoromethyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-5-methyl-N-(oxolan-2-ylmethyl)-2-phenylfuran-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide
(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
ethyl 4-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-phenylbenzamide
[(2,6-difluoro-4-methoxyphenyl)methyl](methyl)(pyrazin-2-ylmethyl)amine
N-(2,4-difluorophenyl)-3-{[methyl(piperidin-3-ylmethyl)amino]methyl}benzamide
4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-3-methylphenol