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4-(cyclohexylmethyl)-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
N,7-dimethyl-N-(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(pyrrolidine-1-carbonyl)piperidine
N-(3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(1H-imidazol-1-yl)propan-1-one
ethyl 3-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)heptanoate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-6-oxo-N-(oxolan-2-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
7-chloro-3-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)methyl]-1,2-dihydroquinolin-2-one
5-cyclobutyl-N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1,3,4-oxadiazol-2-amine
1-[3-(4-fluorophenoxy)azetidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
{4-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]-1,4-oxazepan-6-yl}methanol
5-{[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-N,N-dimethylfuran-2-carboxamide
2,6-dimethyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]quinoline-4-carboxamide
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-3-phenylpropanamide
N-{[5-(quinolin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
2-{4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl}-1,3-benzothiazole
2-ethyl-8-(1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[3-(3-hydroxypiperidin-1-yl)propyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
(2R,6R)-4-(6-hydroxyhexyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3aR,7aS)-2-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
(1S,5R)-3-(oxan-4-yl)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-ethyl-6-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
5-cyclopropanecarbonyl-1'-(5-methyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-amino-4-phenylpyrimidine-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
N-{2-[bis(propan-2-yl)amino]ethyl}-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(morpholin-4-yl)acetamide
3-{[(2E)-3-(furan-2-yl)prop-2-en-1-yl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
N,N,2-trimethyl-7-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
[(3R,4R)-1-(3-fluorobenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-1-(1H-1,3-benzodiazol-2-ylmethyl)-N-ethyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
2-methoxy-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-ethyl-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
(2S)-3-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-ol
4-[(3-ethoxy-2-hydroxypropyl)amino]pyrimidine-5-carboxylic acid
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
2-{4-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyrazine
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-(1H-pyrazol-4-yl)butan-1-one
ethyl 3-(2-phenoxyethyl)-1-propylpiperidine-3-carboxylate
N-cyclopropyl-N-[(3-methoxyphenyl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-(5-benzyl-4-cyclopropanecarbonyl-2-oxopiperazin-1-yl)benzonitrile
3,5-dimethyl-4-{2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-pyrazole
1-methyl-4-(2-methyl-1,3-benzothiazole-5-carbonyl)piperazin-2-one
4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-1,4-diazepan-2-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(2S,4S)-4-amino-1-[(3,5-dichloro-2-methoxyphenyl)methyl]pyrrolidine-2-carboxylic acid