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4-{[5-(hydroxymethyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methyl}-N-(prop-2-en-1-yl)piperidine-1-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(2,3-dimethoxyphenyl)methyl]piperazin-2-one
2-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}butanamide
4-(5-{[1-(2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,4-triazol-3-yl)pyridine
1-tert-butyl-5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
3-[3-({[1-(6-methylpyridin-3-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
(3aR,6aR)-2-methyl-5-[4-(2-oxopyrrolidin-1-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)benzoic acid
3-(1-methyl-1H-pyrazol-4-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)propanamide
8-[3-(1-methoxyethyl)phenyl]quinolin-4-amine
N-[(3R,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-methyl-2-(morpholin-2-yl)-N-[(4-phenoxyphenyl)methyl]acetamide
{4-[(2-cyclohexylpyrimidin-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
1-(4-{1-[(2-chlorophenyl)methyl]-1H-imidazol-2-yl}phenyl)ethan-1-one
2-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}pyridine-3-carboxylic acid
2-{2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
2-[2-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-1-(4-methylpiperidin-1-yl)ethan-1-one
3-{[1-(oxan-4-yl)piperidin-3-yl]formamido}-N-phenylpropanamide
3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-phenylpyrrolidine
N-[(1R,3R)-3-aminocyclopentyl]-4-hydroxy-3-methylbenzamide
2-fluoro-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
methyl (2S)-2-[(1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidin-4-yl)formamido]-2-phenylacetate
2-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxy]-3-(trifluoromethyl)pyridine
(3-{2-[1-(5-fluoropyridine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-(prop-2-en-1-yl)-5-[3-(1H-pyrazol-1-yl)phenyl]furan-2-carboxamide
3-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)pyridin-2-amine
[1-(azepan-1-yl)propan-2-yl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
5-[1-(1-methoxybutan-2-yl)-4-phenyl-1H-imidazol-5-yl]-3-methyl-1,2-benzoxazole
2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-(trimethyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(3,4-difluorophenyl)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
10-methoxy-5-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-(3-methoxypropyl)-3-{2-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
2-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1,2-dihydrophthalazin-1-one
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
(2S)-2-amino-3-cyclohexyl-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
(3S,7S)-5-[2-(morpholin-4-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-phenyl-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-amine
10-methoxy-5-[4-(pyridin-4-yl)pyrimidin-2-yl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[2-(2-methylphenyl)pyrrolidin-1-yl]butan-1-one
N,2-dimethyl-3-phenyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}cycloprop-2-ene-1-carboxamide
N-benzyl-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decane-8-sulfonamide
2-{1-cyclopentyl-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
5-(4-fluorophenyl)-N-(1-methoxybutan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
(3aS,6aS)-2-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid