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(3aS,7aR)-5-methyl-2-(1-methyl-1H-pyrazole-4-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N,2-dimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]imidazo[1,2-a]pyrimidine-3-carboxamide
3-{[3-(adamantan-1-yl)-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[3-(4-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}pyridin-2-yl)phenyl]ethan-1-one
2-amino-4-[2-(2-methylphenyl)pyrimidin-5-yl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
3-(5-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
1-(5-fluoropyrimidin-2-yl)-4-hydroxypiperidine-4-carboxylic acid
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(4-methyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-[4-(3-fluorophenyl)phenyl]-1-{[5-(hydroxymethyl)furan-2-yl]methyl}pyrrolidine-2-carboxamide
7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(3-methylpiperidine-1-carbonyl)quinoline
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,7-dimethyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-methoxy-6-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)phenol
4-[(6-chloropyridin-3-yl)methyl]-2-(3,4-dichlorophenyl)morpholine
3-{1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1-(pyridin-4-yl)ethan-1-ol
2-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyridine
ethyl 4-(cyclopropylmethyl)-1-[2-(trifluoromethoxy)benzenesulfonyl]piperidine-4-carboxylate
(3S,4R)-1-[2-amino-6-(thiophen-2-ylsulfanyl)pyrimidin-4-yl]-4-(hydroxymethyl)piperidin-3-ol
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(3-methoxypropanoyl)piperidine-4-carboxamide
N-phenyl-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}propanamide
1-[1-(furan-2-yl)ethyl]-4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-8-(trifluoromethyl)quinoline
4-({6-[4-(1-methoxyethyl)phenyl]pyridin-3-yl}methyl)morpholine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-4-methoxy-3-(methoxymethyl)benzamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
N2,N2-dimethyl-N4-(3-phenylpropyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-ethyl-N-[(4-fluorophenyl)methyl]-4-hydroxybenzamide
N,N-dimethyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)butanamide
1-(azetidin-1-yl)-2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
2-ethyl-N-[3-(2-methoxyphenyl)propyl]pyrimidine-5-carboxamide
N-[(3S,4R)-1-(2-phenoxybenzoyl)-4-propylpyrrolidin-3-yl]acetamide
2-({4-[4-(2-ethylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
4-[(4-methylphenyl)[2-(thiophen-3-yl)-1H-imidazol-1-yl]methyl]pyridine
methyl 2-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
N-methyl-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}acetamide
(3R,4S)-1-(5-methyl-2-phenylfuran-3-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
2-[3-(propan-2-yl)-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]pyridine
N-cyclopropyl-5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-cyano-1-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrrole-2-carboxamide
3-(2-chlorophenyl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-(methylsulfanyl)-1-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]propan-1-ol
N-(3-cyanophenyl)-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-[3-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenoxy]acetamide
2-[1-(2-methylpropyl)-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
N-[(3R,4S)-1-(cyclobutylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-5-methyl-2H-1,2,3-triazole-4-carboxamide
1-(3-fluoropyridin-4-yl)-4-[(4-methylphenyl)methyl]piperazine
methyl 4-({3-[4-(diethylcarbamoyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)benzoate