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1-[(3-methylphenyl)methyl]-4-(1-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(3-fluorophenoxy)-1-(6-methoxypyrimidin-4-yl)piperidine-4-carboxylic acid
6-(3-fluorophenyl)-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-oxo-1-(2-phenylethyl)-3-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]benzamide
4-{4-[4-(cyclopentylmethyl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-methyl-N-[4-(5-methylfuran-2-amido)phenyl]-1H-pyrazole-5-carboxamide
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-[(1-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperidin-3-yl)methyl]cyclobutanecarboxamide
[(2-tert-butylpyrimidin-5-yl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
2-methyl-N-[2-(pyridin-3-yl)phenyl]propanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-(thiomorpholin-4-yl)ethan-1-one
1-methyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-5-methoxypyridin-4-ol
2-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}-1-(pyrrolidin-1-yl)ethan-1-one
(1S,5R)-N-[(4-fluorophenyl)methyl]-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-({2-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-(2-chloro-4-methylphenyl)-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}propan-1-one
N-(2-{1-[(3-chloro-4-fluorophenyl)methyl]piperidin-2-yl}ethyl)acetamide
1-[1-(4-methylpent-3-en-1-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[(2E)-2-methylbut-2-en-1-yl]amine
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
(1S,3R)-3-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanamido]-N-cyclobutylcyclopentane-1-carboxamide
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidine
2-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N-(propan-2-yl)pyridine-4-carboxamide
2-(2-methoxy-4-methylphenoxymethyl)-4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazole
(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}morpholin-2-yl)methanamine
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
4-(1-methyl-1H-pyrazole-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,3R)-3-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(dimethylamino)ethyl]-4-(quinoxalin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-cyclopropanecarbonyl-4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]piperidine
5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-4-methyl-2-(piperidin-1-yl)pyrimidine
4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
7-(2,3-dimethoxyphenyl)-4-[1-(2-fluorophenyl)propan-2-yl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-(cyclopropylmethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(3-methylthiophen-2-yl)methyl]urea
N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
5-methoxy-9-(3-propyl-1H-pyrazole-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]butanamide
1-{imidazo[1,2-a]pyridine-2-carbonyl}-3-(4-phenoxybenzoyl)piperidine
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[2-(dimethylamino)ethyl]-3-(oxolan-2-ylmethyl)urea
1-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-3-ol