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3-chloro-N-cyclopentyl-4-{[1-(2-methoxyethyl)piperidin-4-yl]oxy}benzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(2-hydroxyethyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
1-(3-oxo-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(5-cyanopyridin-2-yl)-4-{[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}benzamide
1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
5-{4-hydroxy-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-cyclopropylethan-1-one
5-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-acetyl-N-[1-(1-ethyl-1,2,3,6-tetrahydropyridin-4-yl)propan-2-yl]piperidine-4-carboxamide
3-[(3R,4S)-1-[4-(ethylamino)pyrimidin-2-yl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-(2-ethyl-1H-imidazol-1-yl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
N-[3-(1H-indol-1-yl)propyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
N-{1-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-(furan-2-ylmethyl)-3-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]propan-1-ol
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
4-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N'-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]ethanediamide
(2R)-2-amino-3-methyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
(1S,5R)-3-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)urea
N-ethyl-3,5-dimethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1H-pyrazole-4-carboxamide
N-[2-(benzyloxy)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-4-{[(2-chloro-6-fluorophenyl)methyl](ethyl)amino}oxolan-3-ol
4,6-dimethyl-1-(2-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
N,N-dimethyl-5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}pyridin-2-amine
(2,1,3-benzoxadiazol-5-ylmethyl)(4-methoxy-4-methylpentan-2-yl)amine
1-(propane-2-sulfonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(1S,5R)-3-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(4-chlorophenyl)methyl]-8-[3-(1H-imidazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
methyl (2S,4S)-1-[(2-chlorophenyl)methyl]-4-(2,3-dimethyl-1H-indole-7-amido)pyrrolidine-2-carboxylate
5-methyl-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)thiophene-2-carboxamide
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
N-cyclopentyl-1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
N-[2-(furan-2-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
(3S,4S)-1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-cyclopropylpyrrolidine-3-carboxylic acid
4-ethyl-6-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidine
5-(4-fluoro-2-methylphenyl)-1-[3-(1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazole
[(4-ethynylphenyl)methyl]({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
4-(1H-imidazol-1-yl)-1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine-4-carboxylic acid
ethyl 1-(3-acetyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
1-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
1-benzyl-5-(dimethyl-1,2-oxazole-4-carbonyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
1-(azocan-1-yl)-3-(2-methoxy-5-{[(2-phenylethyl)amino]methyl}phenoxy)propan-2-ol
4-[(2,3-difluorophenyl)methyl]-1-(3,5-dimethylphenyl)piperazin-2-one