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N-(butan-2-yl)-3-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-ethylbenzamide
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methyl-1,2-dihydroquinoxalin-2-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(dimethylsulfamoyl)ethyl]benzamide
2-(2-methoxyethyl)-8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
5-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-1,3-oxazole
ethyl 2-{1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]piperidin-2-yl}acetate
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
4-phenoxy-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
4-[(3-{2-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]morpholine
2-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carboxamide
3-{1-[(1-butyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
(4aR,7aS)-4-(3-hydroxybenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-({4-[3-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}methyl)-4-methylpiperazine
3-ethyl-5-methyl-4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,2-oxazole
5-butyl-1'-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-fluoro-2-[2-(1H-imidazol-2-yl)benzoyl]-1-methyl-1,2,3,4-tetrahydroisoquinoline
N,2-dimethyl-6-(piperidin-3-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidin-4-amine
2-{5-[2-(methylsulfanyl)ethyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}-1H-1,3-benzodiazole
4-[3-(3-ethylpiperazine-1-carbonyl)phenyl]-2-methylbutan-2-ol
3-[(2S)-2-amino-4-(methylsulfanyl)butanamido]-N-(2,6-dimethylphenyl)benzamide
(1-{7-ethyl-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-yl)methanol
2-amino-N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3S,4S)-1-(4-methoxybenzoyl)-4-[methyl(oxan-4-ylmethyl)amino]pyrrolidin-3-ol
6-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]quinoline
8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(2-fluorophenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
methyl 4-[2-amino-3-cyano-6-(2,4-dimethylphenyl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
2-(1H-pyrazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
3-[({2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}amino)methyl]pyrrolidin-3-ol
4-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
(1R,5R)-3-cyclobutanecarbonyl-6-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-2-(morpholin-3-yl)acetamide
1-(2-{1-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-chloro-1,3-dimethyl-1H-pyrazole
2-(1-{[1-(5-methylhexan-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
N-{4-[1-ethyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]phenyl}-N-methylmethanesulfonamide
(2S)-1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidine-2-carboxamide
1-[1'-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-tert-butyl-4-hydroxypyrimidine-5-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-2-ethyl-N-(pyridin-2-ylmethyl)butanamide
4-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzonitrile
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]propanamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-aminopyrimidin-5-yl)-7-fluoro-N,N-dimethylquinoline-4-carboxamide
[1-(2-ethylpyrimidin-5-yl)-3-(4-methoxyphenyl)prop-2-yn-1-yl](methyl)(pyrazin-2-ylmethyl)amine
2-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-methyl-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
4-{[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid